SCHEMBL22703003

SCHEMBL22703003

N#Cc1c(N)c2c(c3c1CCc1cc(OCCCCCC(=O)O)ccc1-3)-c1ccc(OCCCCCC=O)cc1CC2

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 7/20 0.38
ITGA2B P08514 7/20 0.38
S1PR1 P21453 2/20 0.38
ALB P02768 1/20 0.37
PPARD Q03181 2/20 0.36
PPARA Q07869 2/20 0.36
FFAR1 O14842 1/20 0.35
PPARG P37231 1/20 0.35
PDK2 Q15119 2/20 0.35
ALK Q9UM73 1/20 0.34
MAOB P27338 3/20 0.33
S1PR3 Q99500 1/20 0.33
EGFR P00533 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20031905 0.93 S1PR1 (0.37) ITGB3ITGA2BS1PR1ALBPPARD
SCHEMBL22683260 0.87 ITGB3 (0.43) ITGB3ITGA2BS1PR1ALBPPARD
SCHEMBL20031911 0.86 MAOB (0.41) ITGB3ITGA2BPPARDPPARAMAOB
SCHEMBL22683257 0.82 MAOB (0.39) ITGB3ITGA2BPPARDPPARAMAOB
SCHEMBL20031639 0.82 ALB (0.44) ITGB3ITGA2BS1PR1ALBPPARD
SCHEMBL20031909 0.82 MAOB (0.43) PPARDPPARAMAOBEGFR
SCHEMBL20031890 0.81 MAOB (0.38) MAOBEGFR
SCHEMBL20031650 0.81 MAOB (0.38) PPARDPPARAMAOBEGFR
SCHEMBL20031904 0.81 THRA (0.43) MAOBEGFR
SCHEMBL22683275 0.79 ITGB3 (0.38) ITGB3ITGA2BS1PR1ALBPPARD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3518746-B1 [5]HELICENE DERIVATIVES AS MOLECULAR REPORTERS FOR DIAGNOSTIC APPLICATIONS AND METHODS OF SYNTHESIS THEREFOR NATIONAL SCIENCE AND TECH DEVELOPMENT AGENCY (TH) 2020-11-25 EP disclosed