SCHEMBL2271237

SCHEMBL2271237

CC(C)(C)OC(=O)c1ccc(CCCCc2ccccc2)cc1NC(=O)c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 12/20 0.48
PLK3 Q9H4B4 6/20 0.48
KDM4E B2RXH2 1/20 0.44
MAPK1 P28482 1/20 0.44
HSD17B10 Q99714 1/20 0.44
HDAC1 Q13547 2/20 0.44
TRPV1 Q8NER1 1/20 0.43
LTC4S Q16873 1/20 0.43
SLC16A3 O15427 1/20 0.43
NR1H4 Q96RI1 1/20 0.43
MCL1 Q07820 1/20 0.43
BCL2A1 Q16548 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2274675 0.98 PLK1 (0.46) PLK1PLK3KDM4EMAPK1HSD17B10
SCHEMBL27716624 0.89 PLK1 (0.47) PLK1PLK3KDM4EMAPK1HSD17B10
SCHEMBL27716638 0.87 HSD17B10 (0.46) PLK1PLK3KDM4EMAPK1HSD17B10
SCHEMBL2273303 0.86 NPC1 (0.43) PLK1PLK3KDM4EMAPK1HSD17B10
SCHEMBL2272564 0.86 ACLY (0.48) HDAC1
SCHEMBL2272409 0.83 PLK1 (0.63) PLK1PLK3HDAC1LTC4SSLC16A3
SCHEMBL2275189 0.82 MAPK1 (0.54) KDM4EMAPK1HSD17B10
SCHEMBL2275549 0.81 SLC16A3 (0.43) PLK1KDM4ESLC16A3
SCHEMBL2270158 0.81 MAPK1 (0.50) KDM4EMAPK1HSD17B10HDAC1NR1H4
SCHEMBL2271236 0.80 PLK1 (0.60) PLK1PLK3HDAC1LTC4SMCL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7999132-B2 Anthranilic acid derivative or salt thereof TOYAMA CHEMICAL CO., LTD. (JP) 2011-08-16 US disclosed
US-20090240052-A1 NOVEL ANTHRANILIC ACID DERIVATIVE OR SALT THEREOF TOYAMA CHEMICAL CO., LTD. (JP) 2009-09-24 US disclosed
EP-1820795-A1 NOVEL ANTHRANILIC ACID DERIVATIVE OR SALT THEREOF TOYAMA CHEMICAL CO., LTD. (JP) 2007-08-22 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090240052-A1 NOVEL ANTHRANILIC ACID DERIVATIVE OR SALT THEREOF MMP13, MMP26, MMP11 PLK1 4227/4885PLK3 3893/4885KDM4E 1257/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.