SCHEMBL22720228

SCHEMBL22720228

COc1nc(C)c(C=O)c(N2CCN(C(=O)OC(C)(C)C)CC2)n1

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TLR9 Q9NR96 2/20 0.42
ALDH1A1 P00352 3/20 0.40
KMT2A Q03164 2/20 0.40
SMPD3 Q9NY59 2/20 0.40
MEN1 O00255 1/20 0.40
RXFP1 Q9HBX9 1/20 0.39
GBA1 P04062 2/20 0.39
CKS1B P61024 2/20 0.39
SKP1 P63208 2/20 0.39
SKP2 Q13309 2/20 0.39
LMNA P02545 1/20 0.38
MAPT P10636 1/20 0.38
MAP4K4 O95819 1/20 0.38
KIT P10721 1/20 0.37
GPR119 Q8TDV5 1/20 0.37
TLR7 Q9NYK1 1/20 0.37
POLB P06746 1/20 0.37
CNR1 P21554 1/20 0.36
CNR2 P34972 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22720236 0.83 TLR9 (0.44) TLR9ALDH1A1KMT2ASMPD3MEN1
SCHEMBL22724587 0.83 TLR9 (0.44) TLR9ALDH1A1KMT2ASMPD3MEN1
SCHEMBL22720272 0.80 KRAS (0.43)
SCHEMBL22720279 0.76 TLR9 (0.43) TLR9ALDH1A1SMPD3GBA1CKS1B
SCHEMBL14697627 0.75 LMNA (0.56) TLR9ALDH1A1KMT2AMEN1GBA1
SCHEMBL21734104 0.74 GBA1 (0.44) TLR9ALDH1A1GBA1CKS1BSKP1
SCHEMBL31651886 0.72 CKS1B (0.48) TLR9ALDH1A1KMT2ASMPD3MEN1
SCHEMBL22873609 0.72 GPR119 (0.55) TLR9ALDH1A1KMT2ASMPD3MEN1
SCHEMBL31652099 0.72 TLR9 (0.54) TLR9SMPD3GBA1CKS1BSKP1
SCHEMBL23560764 0.72 GPR119 (0.50) ALDH1A1KMT2AMEN1GBA1CKS1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113396147-B Aromatic heterocyclic derivative regulator, preparation method and application thereof 上海翰森生物医药科技有限公司 2024-06-18 CN disclosed
CN-112552294-B Piperazine heterocyclic derivative-containing inhibitor, preparation method and application thereof 上海翰森生物医药科技有限公司 2023-12-19 CN disclosed
CN-113396147-A Aromatic heterocyclic derivative regulator, preparation method and application thereof 上海翰森生物医药科技有限公司 2021-09-14 CN disclosed
CN-112552294-A Piperazine heterocyclic derivative inhibitor, preparation method and application thereof 上海翰森生物医药科技有限公司 2021-03-26 CN disclosed
WO-2020239123-A1 AROMATIC HETEROCYCLIC DERIVATIVE MODULATOR AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海翰森生物医药科技有限公司 2020-12-03 WO disclosed