SCHEMBL22723977

SCHEMBL22723977

Cn1ncc(CC(N)=O)c1F

nearest known ligand 0.36

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ICMT O60725 3/20 0.35
HTT P42858 1/20 0.34
P2RX7 Q99572 5/20 0.34
DRD2 P14416 6/20 0.33
DRD3 P35462 6/20 0.33
CFD P00746 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22724157 0.84 DRD3 (0.35) HTTP2RX7DRD2DRD3
SCHEMBL4007505 0.80 HTT (0.39) HTT
SCHEMBL22572506 0.77
SCHEMBL1992512 0.72 RIPK2 (0.39) HTT
SCHEMBL30006444 0.69 LGMN (0.38) ICMTHTTCFD
SCHEMBL25478486 0.68 GABRA1 (0.32)
SCHEMBL22723955 0.68 ICMT (0.37) ICMTHTTDRD2DRD3CFD
SCHEMBL6611651 0.67 MAPT (0.40) HTT
SCHEMBL24828460 0.67 HPGD (0.39) HTT
SCHEMBL1719142 0.67 HPGD (0.48) HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3744721-A1 CONDENSED CYCLIC COMPOUND HAVING DOPAMINE D3 RECEPTOR ANTAGONISM Shionogi & Co., Ltd (JP) 2020-12-02 EP disclosed