SCHEMBL22728397

SCHEMBL22728397

CCC(C#N)(CC)CCc1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 3/20 0.44
DRD3 P35462 3/20 0.44
DRD2 P14416 2/20 0.44
DRD4 P21917 2/20 0.44
LMNA P02545 1/20 0.41
EBP Q15125 3/20 0.40
SIGMAR1 Q99720 3/20 0.40
TP53 P04637 1/20 0.39
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
ALOX15 P16050 1/20 0.38
ALOX12 P18054 1/20 0.38
CASP1 P29466 1/20 0.38
HSD17B10 Q99714 1/20 0.38
ATM Q13315 2/20 0.38
TAAR1 Q96RJ0 3/20 0.38
CHRM2 P08172 1/20 0.37
HTR1A P08908 1/20 0.37
ADRA2A P08913 1/20 0.37
CHRM1 P11229 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22728407 0.91 OPRM1 (0.42) OPRM1DRD3DRD2DRD4EBP
SCHEMBL22728409 0.89 SIGMAR1 (0.43) OPRM1DRD3DRD2DRD4EBP
SCHEMBL2436941 0.78 DRD2 (0.45) OPRM1DRD3DRD2DRD4EBP
SCHEMBL10766520 0.75 TAAR1 (0.45) TP53ALDH1A1HPGDALOX15ALOX12
SCHEMBL11824172 0.75 DRD2 (0.46) OPRM1DRD3DRD2DRD4EBP
SCHEMBL16079189 0.74 DRD2 (0.42) OPRM1DRD3DRD2DRD4EBP
SCHEMBL14477302 0.74 DRD2 (0.46) OPRM1DRD3DRD2DRD4EBP
SCHEMBL11066485 0.72 TP53 (0.44) OPRM1DRD3LMNATP53ALDH1A1
SCHEMBL11224549 0.72 TDP1 (0.50) LMNATP53ALDH1A1HPGDALOX15
SCHEMBL21058275 0.71 TAAR1 (0.45) TP53ALDH1A1HPGDALOX15ALOX12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020243027-A1 COMPOUNDS, COMPOSITIONS, AND METHODS OF USE SAGE THERAPEUTICS, INC. (US) 2020-12-03 WO disclosed