SCHEMBL2273408

SCHEMBL2273408

COc1ccc(CC(O)=S)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.55
HTT P42858 1/20 0.55
PKM P14618 1/20 0.55
CTBP2 P56545 1/20 0.53
LTA4H P09960 1/20 0.52
KDM4E B2RXH2 2/20 0.52
SMN1; SMN2 Q16637 2/20 0.52
MAPT P10636 2/20 0.51
TDP1 Q9NUW8 1/20 0.51
GAA P10253 1/20 0.51
HPGD P15428 1/20 0.51
APOBEC3G Q9HC16 1/20 0.51
IDO1 P14902 1/20 0.50
USP2 O75604 1/20 0.50
TP53 P04637 1/20 0.50
LDHA P00338 1/20 0.50
POLB P06746 1/20 0.50
NPC1 O15118 1/20 0.49
CA12 O43570 1/20 0.48
CA1 P00915 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10969285 0.83 ALDH1A1 (0.55) ALDH1A1HTTPKMCTBP2KDM4E
SCHEMBL5901677 0.81 ALDH1A1 (0.53) ALDH1A1HTTPKMKDM4ESMN1; SMN2
SCHEMBL9564020 0.81 IDO1 (0.54) ALDH1A1HTTPKMCTBP2KDM4E
SCHEMBL7370074 0.80 HTT (0.57) HTTPKMCTBP2LTA4HKDM4E
SCHEMBL498481 0.79 F2RL1 (0.59) ALDH1A1PKMKDM4EPOLBNPC1
SCHEMBL6581234 0.79 LTA4H (0.53) ALDH1A1HTTPKMLTA4HKDM4E
SCHEMBL240822 0.78 KDM4E (0.74) ALDH1A1HTTPKMCTBP2KDM4E
SCHEMBL8134521 0.78 ALDH1A1 (0.50) ALDH1A1HTTPKMCTBP2KDM4E
SCHEMBL18763976 0.78 TAAR1 (0.52) ALDH1A1HTTPKMCTBP2KDM4E
SCHEMBL3665017 0.77 HTT (0.59) ALDH1A1HTTPKMCTBP2LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111808003-A Preparation method of thioether 甘肃农业大学 2020-10-23 CN disclosed
US-9521845-B2 Beta-lactones as antibacterial agents LUDWIG-MAXIMILIANS-UNIVERSITÄT-MÜNCHEN (DE) 2016-12-20 US disclosed
CN-105652595-A Black photosensitive resin composition, black matrix and image display device 东友精细化工有限公司 2016-06-08 CN disclosed
US-20140163094-A1 BETA-LACTONES AS ANTIBACTERIAL AGENTS LUDWIG-MAXIMILIANS-UNIVERSITAT MUNCHEN (DE) 2014-06-12 US disclosed
CN-101434682-B Polymer resin composition SUMITOMO CHEMICAL CO 2014-04-09 CN disclosed
US-8669283-B2 Beta-lactones as antibacterial agents LUDWIG-MAXIMILIANS-UNIVERSITAT MUNCHEN (DE) 2014-03-11 US disclosed
US-8563598-B2 2013-10-22 US disclosed
CN-101121825-B Resin composition capable of polymerizing SUMITOMO CO LTD 2012-07-18 CN disclosed
US-20110196027-A1 BETA-LACTONES AS ANTIBACTERIAL AGENTS LUDWIG-MAXIMILIANS-UNIVERSITAT MUNCHEN 2011-08-11 US disclosed
EP-2254574-A1 BETA-LACTONES AS ANTIBACTERIAL AGENTS Ludwig-Maximilians-Universität München (DE) 2010-12-01 EP disclosed
CN-101735400-A Curable resin composition SUMITOMO CHEMICAL CO 2010-06-16 CN disclosed
WO-2009106211-A1 BETA-LACTONES AS ANTIBACTERIAL AGENTS LUDWIG-MAXIMILIANS-UNIVERSITÄT MÜNCHEN (DE) 2009-09-03 WO disclosed
CN-101434682-A Polymer resin composition SUMITOMO CHEMICAL CO (JP) 2009-05-20 CN disclosed
CN-101121825-A Resin composition capable of polymerizing SUMITOMO CHEMICAL CO (JP) 2008-02-13 CN disclosed
US-4571437-A CATALYTIC HYDROGENATION REDUCTION AND REARRANGEMENT OF NITROBENZENE IN PRESENCE OF SULFUR COMPOUND MALLINCKRODT, INC. (US) 1986-02-18 US disclosed
US-4183951-A PSYCHOTROPIC AGENTS LABORATOIRE L. LAFON (FR) 1980-01-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140163094-A1 BETA-LACTONES AS ANTIBACTERIAL AGENTS ALG8, PGLS, GLA ALDH1A1 4077/4885HTT 2856/4885PKM 3751/4885
US-20110196027-A1 BETA-LACTONES AS ANTIBACTERIAL AGENTS ALG8, PGLS, GLA ALDH1A1 4077/4885HTT 2856/4885PKM 3751/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.