SCHEMBL22748436

SCHEMBL22748436

CCOC(=O)c1c(OC2CCN(C(=O)OC(C)(C)C)C2)c2cc(Cl)c(Cl)cc2n1-c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK8 P45983 3/20 0.46
TP53 P04637 1/20 0.43
POLB P06746 1/20 0.43
NPBWR1 P48145 1/20 0.41
MCHR1 Q99705 1/20 0.41
GPR119 Q8TDV5 1/20 0.40
ALOX15 P16050 1/20 0.40
LMNA P02545 2/20 0.40
ALDH1A1 P00352 2/20 0.40
GAA P10253 2/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
USP30 Q70CQ3 1/20 0.40
PIK3CD O00329 2/20 0.39
PDE4A P27815 1/20 0.39
PDE4B Q07343 1/20 0.39
PDE4C Q08493 1/20 0.39
PDE4D Q08499 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22760191 0.90 MAPK8 (0.46) MAPK8TP53NPBWR1MCHR1GPR119
SCHEMBL22747874 0.86 MAPT (0.43) TP53ALDH1A1GAAMEN1KMT2A
SCHEMBL22760197 0.79 MAPT (0.42) MAPK8TP53ALDH1A1GAAMEN1
SCHEMBL22760106 0.77 MAPK8 (0.49) MAPK8TP53POLBGPR119LMNA
SCHEMBL22760097 0.75 CHRM4 (0.45) MCHR1ALDH1A1MEN1KMT2A
SCHEMBL22760562 0.71 ALDH1A1 (0.67) MAPK8TP53POLBALOX15LMNA
SCHEMBL22760558 0.69 ALDH1A1 (0.52) MAPK8TP53POLBALOX15LMNA
SCHEMBL1769219 0.69 USP30 (0.71) GPR119MEN1KMT2AUSP30PIK3CD
SCHEMBL21409063 0.69 USP30 (0.71) GPR119MEN1KMT2AUSP30PIK3CD
SCHEMBL5153452 0.69 USP30 (0.71) GPR119MEN1KMT2AUSP30PIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020244462-A1 INDOLE DERIVATIVES AND PHARMACEUTICAL USE THEREOF 中国药科大学 2020-12-10 WO disclosed
WO-2020244462-A1 INDOLE DERIVATIVES AND PHARMACEUTICAL USE THEREOF 中国药科大学 2020-12-10 WO disclosed