SCHEMBL22760067

SCHEMBL22760067

CCN(CC)c1c(C(=O)O)n(-c2ccc(OC)cc2)c2cc(Cl)c(Cl)cc12

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
EDNRA P25101 6/20 0.41
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
PPARG P37231 2/20 0.40
MAPK8 P45983 4/20 0.39
RPA1 P27694 1/20 0.38
MAPT P10636 2/20 0.37
MITF O75030 1/20 0.37
ALDH1A1 P00352 1/20 0.37
HTT P42858 1/20 0.37
RAB9A P51151 1/20 0.37
HKDC1 Q2TB90 1/20 0.37
PDE10A Q9Y233 1/20 0.37
EDNRB P24530 1/20 0.37
KDM4E B2RXH2 2/20 0.37
FOLH1 Q04609 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
USP14 P54578 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22747838 0.89 NOTUM (0.42) EDNRAMEN1KMT2AMAPK8ALDH1A1
SCHEMBL22760375 0.87 NOTUM (0.37) MEN1KMT2ARPA1MAPTALDH1A1
SCHEMBL22760346 0.87 FOLH1 (0.45) EDNRAMAPK8MAPTALDH1A1FOLH1
SCHEMBL22760073 0.86 CENPE (0.39) MEN1KMT2APPARGMAPK8FOLH1
SCHEMBL22760373 0.83 FOLH1 (0.36) PPARGMAPK8RPA1KDM4EFOLH1
SCHEMBL22760426 0.82 EDNRA (0.39) EDNRAMEN1KMT2APPARGRPA1
SCHEMBL9538849 0.82 KDM4E (0.57) EDNRAMEN1KMT2APPARGMAPT
SCHEMBL22760140 0.82 NOTUM (0.41) EDNRAMEN1KMT2AMAPK8ALDH1A1
SCHEMBL22760374 0.81 HTT (0.33) HTTFOLH1
SCHEMBL22747843 0.81 MAPK8 (0.40) EDNRAMEN1KMT2APPARGMAPK8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020244462-A1 INDOLE DERIVATIVES AND PHARMACEUTICAL USE THEREOF 中国药科大学 2020-12-10 WO disclosed
CN-112028815-A Indole derivatives and medical application thereof 中国药科大学 2020-12-04 CN disclosed