SCHEMBL22760072

SCHEMBL22760072

CCN(CC)c1c(C(=O)O)n(-c2ccc3c(c2)OCCO3)c2ccc(Cl)c(Cl)c12

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
EDNRA P25101 11/20 0.41
EDNRB P24530 6/20 0.41
HTR2A P28223 6/20 0.39
HTR2C P28335 6/20 0.39
SLC6A4 P31645 6/20 0.39
PTGS1 P23219 1/20 0.36
PTGS2 P35354 1/20 0.36
GLA P06280 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22760066 0.85 EDNRA (0.43) EDNRAEDNRBPTGS1PTGS2
SCHEMBL22760158 0.81 NOTUM (0.41) EDNRAKMT2A
SCHEMBL22760379 0.81 SMN1; SMN2 (0.35) KMT2A
SCHEMBL22760364 0.81 FOLH1 (0.37) EDNRAKMT2A
SCHEMBL22760144 0.81 RPA1 (0.36) EDNRAEDNRBKMT2A
SCHEMBL22747839 0.80 TSHR (0.43) EDNRAEDNRBHTR2AHTR2CSLC6A4
SCHEMBL22747882 0.80 HTT (0.37) KMT2A
SCHEMBL22760068 0.80 CENPE (0.38)
SCHEMBL22760426 0.78 EDNRA (0.39) EDNRAEDNRBKMT2A
SCHEMBL22748255 0.78 NOTUM (0.41) EDNRAEDNRBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020244462-A1 INDOLE DERIVATIVES AND PHARMACEUTICAL USE THEREOF 中国药科大学 2020-12-10 WO disclosed
CN-112028815-A Indole derivatives and medical application thereof 中国药科大学 2020-12-04 CN disclosed