SCHEMBL22760066

SCHEMBL22760066

CCN(CC)c1c(C(=O)O)n(-c2ccc3c(c2)OCCO3)c2cc(Cl)c(Cl)cc12

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
EDNRA P25101 12/20 0.43
EDNRB P24530 6/20 0.43
MAPK8 P45983 1/20 0.39
TSHR P16473 1/20 0.37
PTGS1 P23219 1/20 0.36
PTGS2 P35354 1/20 0.36
HPGD P15428 1/20 0.36
ACACB O00763 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22760072 0.85 EDNRA (0.41) EDNRAEDNRBPTGS1PTGS2
SCHEMBL22760375 0.82 NOTUM (0.37) TSHRSMN1; SMN2
SCHEMBL22760346 0.81 FOLH1 (0.45) EDNRAMAPK8TSHR
SCHEMBL22760073 0.81 CENPE (0.39) MAPK8SMN1; SMN2
SCHEMBL22760140 0.81 NOTUM (0.41) EDNRAMAPK8TSHR
SCHEMBL22760373 0.80 FOLH1 (0.36) MAPK8
SCHEMBL22760067 0.79 EDNRA (0.41) EDNRAEDNRBMAPK8
SCHEMBL22760103 0.78 NPSR1 (0.45) EDNRAEDNRBTSHRHPGDSMN1; SMN2
SCHEMBL22760374 0.78 HTT (0.33) HPGD
SCHEMBL22747838 0.77 NOTUM (0.42) EDNRAEDNRBMAPK8TSHRHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020244462-A1 INDOLE DERIVATIVES AND PHARMACEUTICAL USE THEREOF 中国药科大学 2020-12-10 WO disclosed
CN-112028815-A Indole derivatives and medical application thereof 中国药科大学 2020-12-04 CN disclosed