SCHEMBL22760076

SCHEMBL22760076

O=C(O)c1c(N2CCSCC2)c2c(Cl)c(F)ccc2n1-c1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
EDNRA P25101 2/20 0.38
AKR1C3 P42330 1/20 0.33
MALT1 Q9UDY8 1/20 0.32
FOLH1 Q04609 1/20 0.32
HTT P42858 1/20 0.31
ALDH1A1 P00352 3/20 0.31
HPGD P15428 1/20 0.31
HSD17B10 Q99714 1/20 0.31
LMNA P02545 1/20 0.31
RECQL P46063 1/20 0.31
REN P00797 1/20 0.31
PTGS1 P23219 1/20 0.30
PTGS2 P35354 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22748355 0.90 EDNRA (0.40) EDNRAMALT1FOLH1HTTALDH1A1
SCHEMBL22760063 0.89 EDNRA (0.39) EDNRAMALT1FOLH1ALDH1A1HPGD
SCHEMBL22747830 0.89 EDNRA (0.39) EDNRAMALT1FOLH1ALDH1A1HPGD
SCHEMBL22760496 0.87 REN (0.40) EDNRAHTTALDH1A1HPGDHSD17B10
SCHEMBL22747879 0.87 HPGD (0.42) EDNRAAKR1C3HTTALDH1A1HPGD
SCHEMBL22760091 0.86 KDM4E (0.38) EDNRAMALT1FOLH1ALDH1A1LMNA
SCHEMBL22760100 0.81 SMN1; SMN2 (0.40) EDNRAALDH1A1HPGDHSD17B10
SCHEMBL22760177 0.80 AKR1C3 (0.44) EDNRAAKR1C3HTTALDH1A1HPGD
SCHEMBL22760499 0.80 NOTUM (0.37) EDNRAHTTALDH1A1HPGDHSD17B10
SCHEMBL22760495 0.78 FOLH1 (0.37) EDNRAFOLH1ALDH1A1HPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020244462-A1 INDOLE DERIVATIVES AND PHARMACEUTICAL USE THEREOF 中国药科大学 2020-12-10 WO disclosed