SCHEMBL22760091

SCHEMBL22760091

O=C(O)c1c(N2CCS(=O)(=O)CC2)c2c(Cl)c(F)ccc2n1-c1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.38
EDNRA P25101 1/20 0.37
FAAH O00519 7/20 0.35
SLC6A9 P48067 2/20 0.32
CNR1 P21554 1/20 0.32
CNR2 P34972 1/20 0.32
MALT1 Q9UDY8 1/20 0.31
MAT2A P31153 1/20 0.31
FOLH1 Q04609 1/20 0.31
MAPK8 P45983 2/20 0.31
LMNA P02545 1/20 0.30
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22748355 0.89 EDNRA (0.40) KDM4EEDNRAMALT1FOLH1LMNA
SCHEMBL22760063 0.88 EDNRA (0.39) KDM4EEDNRAMALT1FOLH1LMNA
SCHEMBL22747830 0.88 EDNRA (0.39) KDM4EEDNRAMALT1FOLH1LMNA
SCHEMBL22747879 0.86 HPGD (0.42) KDM4EEDNRAMAT2AMAPK8LMNA
SCHEMBL22760076 0.86 EDNRA (0.38) EDNRAMALT1FOLH1LMNAALDH1A1
SCHEMBL22760496 0.86 REN (0.40) KDM4EEDNRALMNAALDH1A1
SCHEMBL22760100 0.80 SMN1; SMN2 (0.40) KDM4EEDNRAALDH1A1
SCHEMBL22760177 0.79 AKR1C3 (0.44) KDM4EEDNRAMAT2ALMNAALDH1A1
SCHEMBL22760499 0.79 NOTUM (0.37) KDM4EEDNRACNR2LMNAALDH1A1
SCHEMBL22760495 0.77 FOLH1 (0.37) KDM4EEDNRACNR2FOLH1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020244462-A1 INDOLE DERIVATIVES AND PHARMACEUTICAL USE THEREOF 中国药科大学 2020-12-10 WO disclosed