SCHEMBL22760170

SCHEMBL22760170

CCN(CC)c1c(C(=O)OCCNC(C)=O)n(-c2ccccc2)c2ccc(F)c(F)c12

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.36
MAPT P10636 2/20 0.36
GAA P10253 1/20 0.36
MAPK8 P45983 13/20 0.35
MTNR1A P48039 2/20 0.35
MTNR1B P49286 2/20 0.35
HPGD P15428 1/20 0.34
TP53 P04637 1/20 0.34
THRB P10828 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.32
MAPK9 P45984 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22747883 0.86 MAPT (0.50) ALDH1A1MAPTGAAHPGDTP53
SCHEMBL22748263 0.85 MAPK8 (0.40) ALDH1A1MAPTGAAMAPK8HPGD
SCHEMBL22760117 0.81 FOLH1 (0.36) ALDH1A1MAPTGAAMAPK8TP53
SCHEMBL22760451 0.79 LMNA (0.34) ALDH1A1MAPTGAAMAPK8TP53
SCHEMBL22760095 0.77 MAPT (0.48) ALDH1A1MAPTGAAHPGDTP53
SCHEMBL22760414 0.73 EGFR (0.33) MAPTGAA
SCHEMBL22747868 0.71 FOLH1 (0.35) ALDH1A1MAPTGAAMAPK8TP53
SCHEMBL22747829 0.71 FOLH1 (0.35) ALDH1A1MAPTGAAMAPK8TP53
SCHEMBL22760173 0.71 ALDH1A1 (0.53) ALDH1A1MAPTGAAHPGDTP53
SCHEMBL22760085 0.71 EDNRA (0.37) ALDH1A1MAPTGAAMAPK8TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020244462-A1 INDOLE DERIVATIVES AND PHARMACEUTICAL USE THEREOF 中国药科大学 2020-12-10 WO disclosed