SCHEMBL22760403

SCHEMBL22760403

CCOC(=O)c1c(N)c2cc(F)c(Cl)cc2n1Cc1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.46
PIM1 P11309 2/20 0.46
PIM2 Q9P1W9 1/20 0.46
MAPT P10636 3/20 0.46
LMNA P02545 2/20 0.46
KDM4E B2RXH2 2/20 0.46
GAA P10253 2/20 0.46
PKM P14618 1/20 0.46
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
ALDH1A1 P00352 3/20 0.44
POLB P06746 1/20 0.44
ATM Q13315 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
S1PR3 Q99500 4/20 0.44
HPGD P15428 1/20 0.43
CASP1 P29466 1/20 0.43
CASP7 P55210 1/20 0.43
HSD17B10 Q99714 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22760129 0.84 ALDH1A1 (0.50) MAPTKDM4EGAAMEN1KMT2A
SCHEMBL22760408 0.82 PIM1 (0.42) TSHRPIM1PIM2MAPTLMNA
SCHEMBL22760162 0.80 TSHR (0.47) TSHRMAPTLMNAKDM4EGAA
SCHEMBL5214927 0.77 CCR2 (0.59) TSHRMAPTLMNAGAAKMT2A
SCHEMBL22760402 0.77 NOD2 (0.60) TSHRMAPTLMNAKDM4EGAA
SCHEMBL1504118 0.76 MAPT (0.55) TSHRMAPTLMNAKDM4EGAA
SCHEMBL4886339 0.75 PLA2G2A (0.55) TSHRMAPTLMNAKDM4EGAA
SCHEMBL5739057 0.75 KMT2A (0.46) MAPTLMNAKDM4EMEN1KMT2A
SCHEMBL22760543 0.74 ALDH1A1 (0.54) MAPTKDM4EGAAMEN1KMT2A
SCHEMBL6092827 0.74 KMT2A (0.49) MAPTLMNAKDM4EMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020244462-A1 INDOLE DERIVATIVES AND PHARMACEUTICAL USE THEREOF 中国药科大学 2020-12-10 WO disclosed