SCHEMBL22791812

SCHEMBL22791812

Cc1ccc2nc3cc(Cl)ccc3c(Cl)c2c1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.50
POLB P06746 1/20 0.50
HSP90AB1 P08238 1/20 0.48
NR4A2 P43354 1/20 0.47
DHODH Q02127 3/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
MPO P05164 2/20 0.44
ALDH1A1 P00352 2/20 0.44
KDM4E B2RXH2 2/20 0.44
MAPT P10636 1/20 0.44
PKM P14618 1/20 0.43
MAOA P21397 1/20 0.42
MAOB P27338 1/20 0.42
ESR1 P03372 1/20 0.42
ESR2 Q92731 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9595142 0.91 LMNA (0.55) LMNADHODHALDH1A1KDM4EMAPT
SCHEMBL31500251 0.89 MAOA (0.52) POLBNR4A2MPOALDH1A1KDM4E
SCHEMBL9593290 0.87 LMNA (0.62) LMNADHODHMEN1KMT2AALDH1A1
SCHEMBL12047873 0.86 LMNA (0.50) LMNAPOLBHSP90AB1NR4A2DHODH
SCHEMBL20008613 0.83 NR4A2 (0.53) LMNAPOLBHSP90AB1NR4A2KMT2A
SCHEMBL9595057 0.83 NQO2 (0.50) LMNAPOLBNR4A2DHODHKMT2A
SCHEMBL17423119 0.83 POLB (0.55) POLBNR4A2KMT2AMPOALDH1A1
SCHEMBL31500224 0.83 MAOA (0.58) LMNANR4A2MPOALDH1A1KDM4E
SCHEMBL9593843 0.82 LMNA (0.53) LMNADHODHMEN1KMT2AALDH1A1
SCHEMBL27961718 0.82 MAOA (0.67) LMNAMEN1KMT2AALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020248075-A9 TARGETING DNA REPAIR IN TUMOR CELLS VIA INHIBITION OF ERCC1-XPF THE GOVERNORS OF THE UNIVERSITY OF ALBERTA (CA) 2021-10-21 WO disclosed
WO-2020248075-A1 TARGETING DNA REPAIR IN TUMOR CELLS VIA INHIBITION OF ERCC1-XPF THE GOVERNORS OF THE UNIVERSITY OF ALBERTA (CA) 2020-12-17 WO disclosed