SCHEMBL2638776

SCHEMBL2638776

O=C(Nc1ccc(C(F)(F)F)cc1)c1ccccc1C(F)(F)F

nearest known ligand 0.70

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 2/20 0.70
SMN1; SMN2 Q16637 1/20 0.70
NPC1 O15118 1/20 0.66
RAB9A P51151 1/20 0.66
KCNK3 O14649 2/20 0.65
KCNK9 Q9NPC2 2/20 0.65
RXFP1 Q9HBX9 2/20 0.63
PTPRC P08575 1/20 0.60
LMNA P02545 1/20 0.60
GAA P10253 1/20 0.60
AVPR2 P30518 1/20 0.56
GPR27 Q9NS67 1/20 0.56
PTGES O14684 2/20 0.56
EPHX2 P34913 1/20 0.56
TRPV1 Q8NER1 2/20 0.54
F2R P25116 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21652266 0.89 PTGES (0.62) PTGS1SMN1; SMN2NPC1RAB9AKCNK3
SCHEMBL5332281 0.88 KCNK3 (0.75) PTGS1SMN1; SMN2NPC1RAB9AKCNK3
SCHEMBL12334663 0.88 RORC (0.71) PTGS1SMN1; SMN2NPC1RAB9AKCNK3
SCHEMBL21022150 0.87 LMNA (0.66) PTGS1SMN1; SMN2NPC1RAB9AKCNK3
SCHEMBL30791183 0.86 LMNA (0.69) PTGS1SMN1; SMN2NPC1RAB9AKCNK3
SCHEMBL8363754 0.86 KCNK3 (0.64) PTGS1SMN1; SMN2NPC1RAB9AKCNK3
SCHEMBL678924 0.86 PTGS1 (0.72) PTGS1SMN1; SMN2KCNK3KCNK9RXFP1
SCHEMBL96040 0.86 KCNK3 (0.59) PTGS1SMN1; SMN2KCNK3KCNK9RXFP1
SCHEMBL3335567 0.86 KCNK3 (0.59) PTGS1SMN1; SMN2KCNK3KCNK9RXFP1
SCHEMBL20601679 0.84 KCNK3 (0.66) PTGS1SMN1; SMN2NPC1RAB9AKCNK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2011524365-A 2011-09-01 JP claimed
WO-2009152356-A2 COMPOUNDS AND COMPOSITIONS USEFUL FOR THE TREATMENT OF MALARIA IRM LLC (BM) 2009-12-17 WO claimed