SCHEMBL22860752

SCHEMBL22860752

CC(=O)Nc1ccc2nc(Nc3ccc(Cl)c(Cl)c3)c(Nc3ccc(Cl)c(Cl)c3)nc2c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.58
KDM4E B2RXH2 5/20 0.58
MEN1 O00255 5/20 0.58
KMT2A Q03164 5/20 0.58
NPC1 O15118 2/20 0.58
RAB9A P51151 2/20 0.58
PABPC1 P11940 1/20 0.58
EGFR P00533 1/20 0.53
GLA P06280 2/20 0.50
TNNI3 P19429 1/20 0.50
TNNT2 P45379 1/20 0.50
TNNC1 P63316 1/20 0.50
RUNX1 Q01196 1/20 0.50
CBFB Q13951 1/20 0.50
CRHBP P24387 1/20 0.47
CRHR2 Q13324 1/20 0.47
EPHX1 P07099 1/20 0.47
EPHX2 P34913 1/20 0.47
POLB P06746 5/20 0.47
TDP1 Q9NUW8 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29495143 1.00 MAPT (0.58) MAPTKDM4EMEN1KMT2ANPC1
SCHEMBL22860682 0.81 L3MBTL1 (0.52) KDM4EMEN1KMT2ANPC1RAB9A
SCHEMBL29597975 0.81 L3MBTL1 (0.52) KDM4EMEN1KMT2ANPC1RAB9A
SCHEMBL4548035 0.81 EPHX1 (0.70) MAPTKDM4EMEN1KMT2ANPC1
SCHEMBL22860758 0.78 RAB9A (0.71) MAPTKDM4EMEN1KMT2ANPC1
SCHEMBL29598234 0.78 RAB9A (0.71) MAPTKDM4EMEN1KMT2ANPC1
SCHEMBL22860791 0.77 TYMS (0.53) KMT2AEGFRCYP3A4
SCHEMBL29495104 0.77 TYMS (0.53) KMT2AEGFRCYP3A4
SCHEMBL2374293 0.75 MAPT (1.00) MAPTKDM4EMEN1KMT2ANPC1
SCHEMBL9613366 0.75 KDM4E (0.75) MAPTKDM4EMEN1KMT2ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114514229-A Antibacterial and antiparasitic quinoxaline-2, 3-diamine derivatives 阿伯里斯特维斯大学 2022-05-17 CN disclosed
WO-2021001661-A1 ANTIBACTERIAL AND ANTIPARASITIC QUINOXALINE-2,3-DIAMINE DERIVATIVES ABERYSTWYTH UNIVERSITY (GB) 2021-01-07 WO disclosed