SCHEMBL22864003

SCHEMBL22864003

COc1ccc(CN2CCC(C(=O)O)C(C(F)(F)F)C2)cc1

nearest known ligand 0.55

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.52
S1PR5 Q9H228 3/20 0.52
SIGMAR1 Q99720 3/20 0.50
SLC18A3 Q16572 6/20 0.48
DRD2 P14416 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22864002 0.86 KDM4E (0.46) KDM4ESIGMAR1SLC18A3DRD2
SCHEMBL22863936 0.84 S1PR5 (0.70) KDM4ES1PR5SIGMAR1SLC18A3
SCHEMBL6990156 0.77 S1PR5 (0.67) KDM4ES1PR5SIGMAR1SLC18A3
Trifluoroacetic Acid SCHEMBL1921476 0.76 SIGMAR1 (0.55) SIGMAR1
SCHEMBL501146 0.75 S1PR5 (0.54) S1PR5
SCHEMBL501147 0.75 S1PR5 (0.54) S1PR5
SCHEMBL4264860 0.75 S1PR5 (0.54) S1PR5
SCHEMBL27549340 0.75 KDM4E (0.76) KDM4ES1PR5
SCHEMBL28043174 0.74 KDM4E (0.49) KDM4ES1PR5SIGMAR1SLC18A3DRD2
SCHEMBL22488317 0.74 ALDH1A1 (0.57) KDM4ESIGMAR1SLC18A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021003398-A1 INHIBITORS OF LOW MOLECULAR WEIGHT PROTEIN TYROSINE PHOSPHATASE (LMPTP) AND USES THEREOF Sanford Burnham Prebys Medical Discovery Institute (US) 2021-01-07 WO disclosed