SCHEMBL22907692

SCHEMBL22907692

C=C1Cc2cc(C(=C)CSCCCCCCCC)ccc2N1

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 4/20 0.36
ESR2 Q92731 4/20 0.36
EPHX2 P34913 1/20 0.35
CES2 O00748 3/20 0.33
THRB P10828 2/20 0.33
GMNN O75496 1/20 0.33
TP53 P04637 1/20 0.33
POLB P06746 1/20 0.33
MAPT P10636 1/20 0.33
CYP2C9 P11712 1/20 0.33
BLM P54132 1/20 0.33
HSD17B10 Q99714 1/20 0.33
THRA P10827 1/20 0.32
PLA2G4B P0C869 1/20 0.31
FAAH O00519 4/20 0.30
CES1 P23141 4/20 0.30
PLA2G6 O60733 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19985154 0.86 EPHX2 (0.32) EPHX2
SCHEMBL13854238 0.82 EPHX2 (0.46) EPHX2TP53MAPTCYP2C9HSD17B10
SCHEMBL14497589 0.74 EPHX2 (0.58) EPHX2
SCHEMBL17424798 0.70 GMNN (0.49) ESR1ESR2CES2THRBGMNN
SCHEMBL4204194 0.69 EPHX2 (0.61) EPHX2
SCHEMBL29191779 0.68 PLA2G4B (0.41) ESR1ESR2CES2THRBGMNN
SCHEMBL29191780 0.66 MGLL (0.48) CES2THRBGMNNTP53POLB
SCHEMBL19985162 0.65 THRB (0.35) ESR1ESR2CES2THRBGMNN
SCHEMBL17231396 0.64 ALDH1A1 (0.45) EPHX2MAPT
SCHEMBL4198695 0.64 EPHX2 (0.57) EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3142665-B1 MIF INHIBITORS FOR THE ACUTE OR CHRONIC TREATMENT OF PULMONARY HYPERTENSION APAXEN (BE) 2021-01-20 EP disclosed