SCHEMBL22908555

SCHEMBL22908555

CC#Cc1cc(Cl)c(C2C(=O)CC3(CCN(C(=O)c4cccnn4)CC3)CC2=O)c(OC)c1

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CCR8 P51685 6/20 0.36
KCNH2 Q12809 6/20 0.36
NAMPT P43490 1/20 0.34
CYP3A4 P08684 6/20 0.33
CYP2D6 P10635 5/20 0.33
HTR1A P08908 2/20 0.33
DRD2 P14416 2/20 0.33
ADRA1A P35348 2/20 0.33
USP2 O75604 2/20 0.33
NSD2 O96028 2/20 0.33
ACACA Q13085 1/20 0.33
HTR4 Q13639 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22908539 0.89 CCR8 (0.47) CCR8KCNH2CYP3A4CYP2D6DRD2
SCHEMBL22908445 0.89 CYP3A4 (0.34) CCR8KCNH2CYP3A4CYP2D6HTR1A
SCHEMBL22908439 0.87 HTR1A (0.38) CCR8KCNH2HTR1AACACA
SCHEMBL22908552 0.86 CYP3A4 (0.44) CCR8KCNH2CYP3A4CYP2D6USP2
SCHEMBL22992042 0.86 NAMPT (0.37) CCR8KCNH2NAMPTCYP3A4CYP2D6
SCHEMBL22908553 0.85 TDP1 (0.43) CCR8KCNH2CYP3A4CYP2D6
SCHEMBL22908440 0.85 HTR1A (0.37) CCR8KCNH2CYP3A4CYP2D6HTR1A
SCHEMBL22908538 0.85 CCR8 (0.41) CCR8KCNH2CYP3A4CYP2D6HTR1A
SCHEMBL22908432 0.85 ACACA (0.33) CCR8KCNH2ACACA
SCHEMBL22908441 0.84 DRD3 (0.41) CCR8KCNH2HTR1AADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021009048-A1 HERBICIDAL CYCLOHEXANEDIONE DERIVATIVES SYNGENTA CROP PROTECTION AG (CH) 2021-01-21 WO disclosed