SCHEMBL22955477

SCHEMBL22955477

CN1CCN(C(=O)c2ccc3[nH]c(-c4cccc5ccccc45)nc3c2)CC1

nearest known ligand 0.55

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDR P35968 3/20 0.55
FGFR1 P11362 2/20 0.55
PDGFRB P09619 1/20 0.55
HPGD P15428 1/20 0.52
TSHR P16473 1/20 0.52
KDM4E B2RXH2 1/20 0.50
ALDH1A1 P00352 1/20 0.50
MAPT P10636 1/20 0.50
HTR2C P28335 1/20 0.49
HRH4 Q9H3N8 2/20 0.48
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
BTK Q06187 3/20 0.45
FLT1 P17948 1/20 0.45
MGLL Q99685 1/20 0.45
TLR9 Q9NR96 1/20 0.44
TLR8 Q9NR97 1/20 0.44
TLR7 Q9NYK1 1/20 0.44
ADORA2A P29274 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22955526 0.92 KDR (0.65) KDRFGFR1PDGFRBHPGDTSHR
SCHEMBL22955364 0.89 HPGD (0.55) HPGDKDM4EALDH1A1MAPTHTR2C
SCHEMBL22955351 0.88 MEN1 (0.59) HPGDKDM4EHTR2CMEN1KMT2A
SCHEMBL22955525 0.88 KDR (0.42) KDRFGFR1PDGFRBHPGDTSHR
SCHEMBL20765466 0.84 ALDH1A1 (0.64) KDRFGFR1PDGFRBHPGDTSHR
SCHEMBL5952108 0.82 FGFR1 (0.58) KDRFGFR1PDGFRBHPGDTSHR
SCHEMBL22955692 0.81 MGLL (0.53) KDRFGFR1PDGFRBHPGDALDH1A1
SCHEMBL2310280 0.80 KDR (0.50) KDRFGFR1PDGFRBHPGDTSHR
SCHEMBL13042446 0.80 KDR (0.58) KDRFGFR1PDGFRBHPGDTSHR
SCHEMBL22955686 0.80 RAB9A (0.53) HPGDKDM4EALDH1A1MAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021022061-A1 ARYL HYDROCARBON RECEPTOR ACTIVATORS OREGON STATE UNIVERSITY (US) 2021-02-04 WO disclosed