Transtorine

Transtorine

SCHEMBL22979

O=C(O)c1cc(O)c2ccccc2n1

nearest known ligand 0.60

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 3/20 0.60
MGAM O43451 1/20 0.53
ALDH1A1 P00352 3/20 0.52
HPGD P15428 1/20 0.52
HSD17B10 Q99714 1/20 0.52
THRB P10828 1/20 0.47
PDE10A Q9Y233 3/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
KDM4E B2RXH2 2/20 0.46
LMNA P02545 1/20 0.46
MYC P01106 1/20 0.46
MAX P61244 1/20 0.46
IGFBP3 P17936 2/20 0.46
MAPT P10636 1/20 0.45
POLB P06746 1/20 0.45
DHODH Q02127 2/20 0.45
IGFBP5 P24593 1/20 0.44
TSHR P16473 1/20 0.43
ACMSD Q8TDX5 1/20 0.43
TDP1 Q9NUW8 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Transtorine SCHEMBL17596601 1.00 ALOX15 (0.60) ALOX15MGAMALDH1A1HPGDHSD17B10
Transtorine SCHEMBL1421892 0.98 ALOX15 (0.58) ALOX15MGAMALDH1A1HPGDHSD17B10
Transtorine SCHEMBL480985 0.98 ALOX15 (0.58) ALOX15MGAMALDH1A1HPGDHSD17B10
Transtorine SCHEMBL21384236 0.86 ALOX15 (0.48) ALOX15MGAMALDH1A1HPGDHSD17B10
SCHEMBL247555 0.85 GRM2 (0.59) ALDH1A1
SCHEMBL17718271 0.85 ALDH1A1 (0.49) ALOX15MGAMALDH1A1HPGDHSD17B10
Transtorine SCHEMBL10895515 0.84 G6PD (0.59) ALOX15ALDH1A1HPGDTHRBPDE10A
Transtorine SCHEMBL7937597 0.84 ALDH1A1 (0.44) ALOX15MGAMALDH1A1HPGDHSD17B10
Hydrochloric Acid SCHEMBL17769122 0.84 GRM2 (0.57) ALDH1A1
SCHEMBL11827386 0.82 IGFBP5 (0.47) ALOX15MGAMALDH1A1HPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 6045 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260146967-A1 DEVICE AND SENSOR FOR DETECTION OF AN ANALYTE REMINDED, INC. (US) 2026-05-28 US claimed
US-20260108550-A1 NICOTINAMIDE MONONUCLEOTIDE DERIVATIVES AND USE THEREOF IN THE TREATMENT AND PREVENTION OF A RED BLOOD CELL DISORDER NUVAMID SA (CH) 2026-04-23 US claimed
US-20260096574-A1 CHOCOLATE REPLICAS PRODUCED FROM INDIVIDUAL COMPONENTS VOYAGE FOODS INC (US) 2026-04-09 US claimed
EP-4405047-B1 CANNABINOID FORMULATION FOR ORAL ADMINISTRATION CB21 PHARMA S R O (CZ) 2026-04-01 EP claimed
EP-4072319-B1 COMPOSITIONS FOR USE IN THE REDUCTION OF NOCICEPTION AND OTHER HEALTH BENEFITS IN INFANTS AND YOUNG CHILDREN NESTLE SA (CH) 2026-04-01 EP claimed
US-20260076956-A1 METHODS FOR REGRESSING OR REVERSING FIBROSIS AND/OR LIVER CIRRHOSIS IN A SUBJECT IN NEED THEREOF USING HIGH-DOSE NIACIN, OR A NIACIN ANALOG THEREOF US GOV VETERANS AFFAIRS (US) 2026-03-19 US claimed
US-12551459-B2 Combination of kynurenine and antigen presenting cells (APC) as therapeutics and methods for their use in immune modulation THE UNIVERSITY OF BRITISH COLUMBIA (CA) 2026-02-17 US claimed
US-20260007144-A1 CHOCOLATE REPLICAS PRODUCED FROM INDIVIDUAL COMPONENTS VOYAGE FOODS INC (US) 2026-01-08 US claimed
US-20250367192-A1 BICYCLIC COMPOUNDS AND METHODS FOR THEIR USE IN TREATING PITT HOPKINS SYNDROME NEUREN PHARMACEUTICALS LTD (NZ) 2025-12-04 US claimed
EP-4648788-A1 LIPID BINDING PROTEIN MOLECULE THERAPY Abionyx Pharma SA (FR) 2025-11-19 EP claimed
WO-1995003815-A1 ANTIBODIES SPECIFIC TO QUINOLINIC ACID GEORGETOWN UNIVERSITY (US) 1995-02-09 WO claimed
EP-0564676-A1 Light polarizing material based on quinaldic acid derivatives RESEARCH FRONTIERS INCORPORATED (US) 1993-10-13 EP claimed
EP-0321516-B1 3-INDOLEPYRUVIC ACID DERIVATIVES AND PHARMACEUTICAL USE THEREOF POLIFARMA S.p.A. (IT) 1993-03-03 EP claimed
US-5039528-A EAA antagonists as anti-emetic drugs OLNEY JOHN W (US) 1991-08-13 US claimed
EP-0432994-A2 Excitatory amino acid antagonists as anti-emetic drugs Olney, John William (US) 1991-06-19 EP claimed
EP-0421946-A2 3-indolepyruvic acid derivatives their method of production and therapeutic use POLIFARMA S.p.A. (IT) 1991-04-10 EP claimed
WO-1988007851-A1 LIPOSOME ENTRAPPED N-METHYL-D-ASPARTATE RECEPTOR BLOCKERS INNOVATIVE THERAPEUTICS CORPORATION (US) 1988-10-20 WO claimed
US-4620850-A HYDROXYBENZOLFURANONE WELLA AKTIENGESELLSCHAFT (DE) 1986-11-04 US claimed
EP-0026474-B1 COMPOSITION AND PROCESS FOR OXIDATIVE DYEING OF HAIR Wella Aktiengesellschaft (DE) 1983-06-08 EP claimed
EP-0026473-B1 OXIDATIVE HAIR-DYEING COMPOSITION Wella Aktiengesellschaft (DE) 1983-05-25 EP claimed