SCHEMBL22979591

SCHEMBL22979591

C[C@H](Cc1cn2nccc2nc1Cl)NC(=O)O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.35
RAB9A P51151 3/20 0.35
KIT P10721 2/20 0.34
PCSK9 Q8NBP7 1/20 0.34
DDR1 Q08345 1/20 0.34
ACACB O00763 2/20 0.33
CBLB Q13191 1/20 0.33
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
ESR1 P03372 1/20 0.32
KCNH2 Q12809 1/20 0.32
KCNN3 Q9UGI6 1/20 0.32
LMNA P02545 2/20 0.32
ALDH1A1 P00352 1/20 0.31
CYP2C19 P33261 1/20 0.31
HTT P42858 1/20 0.31
TAAR1 Q96RJ0 1/20 0.31
SCD O00767 1/20 0.31
SCD5 Q86SK9 1/20 0.31
TP53 P04637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22979593 1.00 NPC1 (0.35) NPC1RAB9AKITPCSK9DDR1
SCHEMBL22996558 0.84 PCSK9 (0.48) PCSK9MEN1KMT2ALMNAALDH1A1
SCHEMBL22996562 0.78 KMT2A (0.35) KMT2ATAAR1
SCHEMBL22979871 0.76 KCNN3 (0.36) NPC1RAB9ACBLBKCNN3ALDH1A1
SCHEMBL22979868 0.76 KCNN3 (0.36) NPC1RAB9ACBLBKCNN3ALDH1A1
SCHEMBL18422575 0.68 LMNA (0.50) NPC1RAB9AESR1KCNH2LMNA
SCHEMBL22978874 0.68 PDE10A (0.32) KMT2AKCNN3
SCHEMBL22996432 0.66 SIRT2 (0.31)
SCHEMBL24253457 0.64 GABRA1 (0.35) KITPCSK9DDR1ESR1KCNN3
SCHEMBL4333892 0.63 NPC1 (0.49) NPC1RAB9AMEN1KMT2AESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021027503-A1 TRICYCLIC COMPOUND, PREPARATION METHOD THEREFOR, AND INTERMEDIATE AND USE THEREOF 罗欣药业(上海)有限公司 2021-02-18 WO disclosed