SCHEMBL22982373

SCHEMBL22982373

O=C(O)N1CCc2ccc(CCl)c(F)c2C1

nearest known ligand 0.36

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PNMT P11086 14/20 0.36
ESR1 P03372 2/20 0.34
ESR2 Q92731 2/20 0.34
HTR5A P47898 1/20 0.33
ERCC1 P07992 1/20 0.33
ERCC4 Q92889 1/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.33
ABHD6 Q9BV23 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22981745 0.87 NPC1 (0.35) ESR1ESR2HTR5APTGDR2ABHD6
SCHEMBL22993222 0.81 ESR2 (0.52) ESR2ABHD6
SCHEMBL29697629 0.81 ESR2 (0.52) ESR2ABHD6
SCHEMBL29388817 0.81 ESR2 (0.52) ESR2ABHD6
SCHEMBL22982829 0.76 PNMT (0.37) PNMTESR1ESR2ERCC1ERCC4
SCHEMBL29097985 0.74 DRD2 (0.48) PNMTESR1ESR2
SCHEMBL22981196 0.72 ESR1 (0.43) ESR1ESR2
SCHEMBL22981751 0.72 BTK (0.34) ESR1ESR2HTR5AERCC1ERCC4
SCHEMBL13082467 0.72 RIPK1 (0.49) HTR5APTGDR2ABHD6
SCHEMBL16147790 0.70 TMEM97 (0.41) HTR5APTGDR2ABHD6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4010333-A1 PLASMA KALLIKREIN INHIBITORS Kalvista Pharmaceuticals Limited (GB) 2022-06-15 EP disclosed
WO-2021028645-A1 PLASMA KALLIKREIN INHIBITORS KALVISTA PHARMACEUTICALS LIMITED (GB) 2021-02-18 WO disclosed
WO-2021028649-A1 PLASMA KALLIKREIN INHIBITORS KALVISTA PHARMACEUTICALS LIMITED (GB) 2021-02-18 WO disclosed