SCHEMBL22995089

SCHEMBL22995089

COc1cc(C(C)NC(C)=O)ncc1F

nearest known ligand 0.46

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.40
ROCK2 O75116 7/20 0.39
ROCK1 Q13464 6/20 0.39
ACACB O00763 3/20 0.39
ACACA Q13085 2/20 0.38
BRAF P15056 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22990322 1.00 L3MBTL1 (0.40) L3MBTL1ROCK2ROCK1ACACBACACA
SCHEMBL22995195 0.85 CACNA1I (0.40)
SCHEMBL22990325 0.81 EGFR (0.35) ROCK2ROCK1
SCHEMBL22978636 0.77 P2RX3 (0.37)
SCHEMBL30525606 0.77 P2RX3 (0.37)
SCHEMBL21859435 0.76 P2RX3 (0.41)
SCHEMBL22978515 0.73 P2RX3 (0.37)
SCHEMBL4566147 0.72 CACNA1I (0.60) ACACBACACA
SCHEMBL588472 0.71 APLNR (0.48) L3MBTL1ACACBACACA
SCHEMBL12069877 0.71 APLNR (0.48) L3MBTL1ACACBACACA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021028806-A1 HETEROCYCLIC WDR5 INHIBITORS AS ANTI-CANCER COMPOUNDS NOVARTIS AG (CH) 2021-02-18 WO disclosed