SCHEMBL27664005

SCHEMBL27664005

COC(=O)C(c1ccccc1)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.51
ACP3 P15309 1/20 0.51
TACR1 P25103 5/20 0.51
LDHB P07195 2/20 0.51
LDHA P00338 1/20 0.51
PTPN1 P18031 1/20 0.49
CNR2 P34972 1/20 0.48
NOS3 P29474 1/20 0.46
NOS1 P29475 1/20 0.46
NOS2 P35228 1/20 0.46
CES2 O00748 1/20 0.46
CES1 P23141 1/20 0.46
NR1H2 P55055 1/20 0.45
NR1H3 Q13133 1/20 0.45
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
PDPK1 O15530 1/20 0.44
CASR P41180 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1578804 0.84 KMT2A (0.69) KMT2A
SCHEMBL2304585 0.81 ACP3 (0.56) ACP3TACR1PTPN1CNR2CES2
SCHEMBL27683652 0.81 ACP3 (0.59) ACP3TACR1LDHBLDHAPTPN1
SCHEMBL27690530 0.81 L3MBTL1 (0.47) KMT2ATACR1
SCHEMBL16781996 0.80 PTPN1 (0.72) ACP3TACR1LDHBLDHAPTPN1
SCHEMBL27965719 0.80 CES2 (0.45) KMT2AACP3TACR1CES2
SCHEMBL6809648 0.80 ALDH1A1 (0.51) LDHBLDHACNR2NOS3NOS1
SCHEMBL28093888 0.80 KMT2A (0.58) KMT2ACNR2
SCHEMBL2843638 0.80 KMT2A (0.58) KMT2ACNR2
SCHEMBL840978 0.79 LDHB (0.50) KMT2AACP3LDHBLDHACNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1993120-B Arylacetic acids and related compounds for treatment of alzheimer's disease MERCK SHARP & DOHME BLURTON PETER 2010-05-05 CN disclosed
CN-1993120-A Arylacetic acids and related compounds for treatment of alzheimer's disease MERCK SHARP & DOHME BLURTON PE (GB) 2007-07-04 CN disclosed