SCHEMBL23074751

SCHEMBL23074751

CCc1ccnc(C)c1C(F)(F)F

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.33
GAA P10253 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
NOS3 P29474 1/20 0.32
NOS2 P35228 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
PSEN1 P49768 1/20 0.32
PSEN2 P49810 1/20 0.32
APH1B Q8WW43 1/20 0.32
NCSTN Q92542 1/20 0.32
APH1A Q96BI3 1/20 0.32
PSENEN Q9NZ42 1/20 0.32
TACR1 P25103 2/20 0.31
HRH4 Q9H3N8 2/20 0.31
PTGS2 P35354 4/20 0.31
MAOA P21397 1/20 0.31
LOXL2 Q9Y4K0 1/20 0.31
KDM4E B2RXH2 1/20 0.31
CYP2A6 P11509 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21181757 0.79 NOTUM (0.32) ALDH1A1GAAL3MBTL1LOXL2KDM4E
SCHEMBL25786516 0.79 RXRA (0.31)
SCHEMBL17002575 0.75 CCR1 (0.38) NOS3NOS2MAOALOXL2CYP2A6
SCHEMBL17531150 0.74 HPGD (0.43) ALDH1A1GAAL3MBTL1KDM4ESYK
Ammonia Solution, Strong SCHEMBL28037175 0.74 CCR1 (0.37) NOS3NOS2MAOACYP2A6
SCHEMBL23193106 0.74 GABRA1 (0.48) ALDH1A1NOS3NOS2KDM4ECYP2A6
SCHEMBL20347074 0.74 TRPV4 (0.34) NOS3NOS2MAOACYP2A6
SCHEMBL11970836 0.74 NOS3 (0.35) NOS3NOS2HRH4CYP2A6
SCHEMBL3801869 0.73 NOS2 (0.38) NOS3NOS2CYP2A6GABRA1GABRB2
SCHEMBL13256363 0.72 GABRA1 (0.46) ALDH1A1GAAPTGS2KDM4EGABRA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021043322-A1 AZEPINO PYRIMIDINE DERIVATIVES AND MEDICAL USE THEREOF 正大天晴药业集团南京顺欣制药有限公司 2021-03-11 WO disclosed