SCHEMBL2312288

SCHEMBL2312288

Cc1c(C(=O)NCCCc2ccccc2)c2ccccc2c(=O)n1Cc1ccoc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 4/20 0.51
TDP1 Q9NUW8 1/20 0.51
TSHR P16473 1/20 0.48
MEN1 O00255 5/20 0.45
KMT2A Q03164 5/20 0.45
POLB P06746 2/20 0.45
USP2 O75604 1/20 0.45
GAA P10253 1/20 0.45
KDM4E B2RXH2 2/20 0.43
HPGD P15428 2/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
LMNA P02545 1/20 0.43
ALOX15 P16050 1/20 0.43
MAPK1 P28482 1/20 0.43
HTT P42858 1/20 0.43
HSD17B10 Q99714 1/20 0.43
ALDH1A1 P00352 1/20 0.42
GFER P55789 1/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3344869 0.82 LMNA (0.43) TSHRMEN1KMT2APOLBGAA
SCHEMBL1365646 0.78 PPARG (0.44) TSHRMEN1KMT2ASMN1; SMN2MAPK1
SCHEMBL2313394 0.75 L3MBTL1 (0.54) L3MBTL1TDP1TSHRMEN1KMT2A
SCHEMBL2149158 0.72 L3MBTL1 (0.51) L3MBTL1TDP1TSHRMEN1KMT2A
SCHEMBL3350444 0.71 SMN1; SMN2 (0.58) TSHRMEN1KMT2APOLBKDM4E
SCHEMBL2313628 0.68 HTR2A (0.36) L3MBTL1TSHRMEN1KMT2APOLB
SCHEMBL1366629 0.67 PPARG (0.52) TSHRMEN1KMT2ASMN1; SMN2MAPK1
SCHEMBL15969988 0.66 L3MBTL1 (0.83) L3MBTL1TDP1MEN1KMT2AKDM4E
SCHEMBL164622 0.63 L3MBTL1 (0.72) L3MBTL1TSHRKMT2APOLBGAA
SCHEMBL1940351 0.63 PTGDR2 (0.75)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2350015-A1 ISOQUINOLINONE DERIVATIVES AS NK3 ANTAGONISTS H. Lundbeck A/S (DK) 2011-08-03 EP claimed