SCHEMBL2312930

SCHEMBL2312930

Nc1nccc(OC(=O)O)n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NUDT1 P36639 2/20 0.47
HSP90AA1 P07900 2/20 0.40
AURKA O14965 1/20 0.40
PRKACA P17612 1/20 0.40
ADORA2A P29274 1/20 0.40
ROCK1 Q13464 5/20 0.39
ALOX5AP P20292 1/20 0.38
FEN1 P39748 1/20 0.38
BCL6 P41182 1/20 0.37
KDR P35968 2/20 0.36
GABRP O00591 1/20 0.36
GABRD O14764 1/20 0.36
GABRA1 P14867 1/20 0.36
GABRB1 P18505 1/20 0.36
GABRG2 P18507 1/20 0.36
GABRB3 P28472 1/20 0.36
GABRA5 P31644 1/20 0.36
GABRA3 P34903 1/20 0.36
GABRA2 P47869 1/20 0.36
GABRB2 P47870 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1505810 0.80 LMNA (0.37) HSP90AA1GABRPGABRDGABRA1GABRB1
SCHEMBL27638894 0.79 NUDT1 (0.50) NUDT1ROCK1HRH4CDC7
SCHEMBL686891 0.78 MAPT (0.33) HSP90AA1HDAC6POLB
SCHEMBL9565270 0.78 PLAAT3 (0.37) HDAC6POLB
Bromide SCHEMBL5348109 0.78 NUDT1 (0.49) NUDT1HSP90AA1AURKAPRKACAADORA2A
SCHEMBL8393570 0.77 SORT1 (0.37) GRM4HDAC6
SCHEMBL11212136 0.74 NUDT1 (0.57) NUDT1HSP90AA1AURKAPRKACAADORA2A
SCHEMBL1885320 0.74 NUDT1 (0.46) NUDT1HSP90AA1AURKAPRKACAADORA2A
SCHEMBL11303883 0.73
SCHEMBL686300 0.73 KMT2A (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1888579-B1 NOVEL FLUORENE DERIVATIVES, COMPOSITION CONTAINING SAID DERIVATIVES AND THE USE THEREOF AVENTIS PHARMA SA (FR) 2011-08-03 EP claimed
EP-3083586-B1 NOVEL CARBOXAMIDES, METHOD FOR THE PRODUCTION THEREOF, PHARMACEUTICAL PREPARATIONS COMPRISING THEM, AND USE THEREOF FOR PRODUCING MEDICAMENTS Bayer Pharma AG (DE) 2018-04-18 EP disclosed
EP-0511072-A1 2-Aminopyrimidin-4-carboxamid derivatives, their preparation and their therapeutical use SYNTHELABO (FR) 1992-10-28 EP disclosed