SCHEMBL23154100

SCHEMBL23154100

C=C(CC)N1CCN(c2cccnc2)CC1

nearest known ligand 0.59

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 2/20 0.49
CHRNA4 P43681 2/20 0.49
HRH3 Q9Y5N1 3/20 0.47
ADAMTS5 Q9UNA0 2/20 0.47
PHGDH O43175 1/20 0.47
TRPV1 Q8NER1 1/20 0.46
GPR119 Q8TDV5 1/20 0.44
ALDH1A1 P00352 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21163168 0.84 GPR119 (0.47) CHRNB2CHRNA4HRH3ADAMTS5PHGDH
SCHEMBL19001331 0.84 ADAMTS5 (0.58) CHRNB2CHRNA4HRH3ADAMTS5TRPV1
SCHEMBL9557965 0.79 CHRNB2 (0.59) CHRNB2CHRNA4TRPV1
SCHEMBL30663952 0.78 TRPV1 (0.54) CHRNB2CHRNA4HRH3ADAMTS5TRPV1
SCHEMBL1433477 0.78 TRPV1 (0.54) CHRNB2CHRNA4HRH3ADAMTS5TRPV1
SCHEMBL27781454 0.78 TRPV1 (0.56) CHRNB2CHRNA4ADAMTS5TRPV1GPR119
SCHEMBL6888784 0.78 CHRNA7 (0.62) CHRNB2CHRNA4HRH3
SCHEMBL29352658 0.78 CHRNA7 (0.62) CHRNB2CHRNA4HRH3
SCHEMBL1981285 0.76 TRPV1 (0.55) CHRNB2CHRNA4ADAMTS5TRPV1GPR119
SCHEMBL25645426 0.75 ALDH1A1 (0.50) HRH3ADAMTS5ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021057882-A1 EGFR INHIBITOR, COMPOSITION AND PREPARATION METHOD THEREFOR 贝达药业股份有限公司 2021-04-01 WO disclosed