SCHEMBL2316362

SCHEMBL2316362

CC(=O)CCC1=CC(C)(C)COc2ccc(C)cc21

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 0.34
SLC6A2 P23975 1/20 0.34
HTR2C P28335 1/20 0.34
HTR2B P41595 1/20 0.34
SIGMAR1 Q99720 1/20 0.34
MEN1 O00255 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2C9 P11712 1/20 0.34
KMT2A Q03164 1/20 0.34
L3MBTL1 Q9Y468 3/20 0.34
KDM4E B2RXH2 4/20 0.33
PKM P14618 2/20 0.33
CTNNB1 P35222 2/20 0.33
WNT3A P56704 2/20 0.33
ALDH1A1 P00352 1/20 0.33
RECQL P46063 1/20 0.33
MAPK1 P28482 2/20 0.33
HTT P42858 2/20 0.33
LMNA P02545 1/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2314396 0.86 MAPT (0.34) MEN1CYP1A2CYP2C9KMT2AL3MBTL1
SCHEMBL2319689 0.86 NOTUM (0.34) MEN1KMT2AHTTMAPTSMN1; SMN2
SCHEMBL2322133 0.86 ALDH1A1 (0.39) L3MBTL1KDM4ECTNNB1WNT3AALDH1A1
SCHEMBL2314339 0.85 PARP1 (0.38) SLC6A2MEN1CYP1A2KMT2AKDM4E
SCHEMBL2321527 0.85 IMPDH2 (0.31)
SCHEMBL2319253 0.84 KDM4E (0.43) HTR1ASLC6A2HTR2BSIGMAR1CYP1A2
SCHEMBL2320678 0.84 MEN1 (0.33) MEN1KMT2APKMHPGD
SCHEMBL2316423 0.81 BACE1 (0.38) CYP2C9HPGDSMN1; SMN2
SCHEMBL2319041 0.79 CYP3A4 (0.35) HTR1ASLC6A2HTR2CHTR2BSIGMAR1
SCHEMBL2317591 0.77 CYP3A4 (0.43) HTR1ASLC6A2HTR2BSIGMAR1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1609786-B1 5-alkenone-3,3-dimethyl-benzoxepines derivatives useful for the preparation of antidiabetic pentadienoic acids MERCK SANTE SAS (FR) 2011-08-03 EP claimed