SCHEMBL2322133

SCHEMBL2322133

CC(=O)CCC1=CC(C)(C)COc2ccc(F)cc21

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.39
KDM4E B2RXH2 2/20 0.39
GAA P10253 2/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
NOTUM Q6P988 1/20 0.34
DRD2 P14416 1/20 0.34
FABP6 P51161 1/20 0.34
AKR1B1 P15121 4/20 0.34
KIF11 P52732 2/20 0.34
PGR P06401 2/20 0.33
NR3C2 P08235 1/20 0.33
AR P10275 1/20 0.33
CTNNB1 P35222 3/20 0.33
CYP19A1 P11511 1/20 0.32
HPGD P15428 1/20 0.31
WNT3A P56704 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2316362 0.86 HTR1A (0.34) ALDH1A1KDM4EL3MBTL1PGRCTNNB1
SCHEMBL2319689 0.85 NOTUM (0.34) NOTUMAKR1B1PGRARCYP19A1
SCHEMBL2314396 0.85 MAPT (0.34) ALDH1A1KDM4EL3MBTL1AKR1B1PGR
SCHEMBL2314339 0.84 PARP1 (0.38) ALDH1A1KDM4EGAAHPGD
SCHEMBL2316043 0.84 HDAC1 (0.34) PGR
SCHEMBL2319253 0.83 KDM4E (0.43) ALDH1A1KDM4EGAAPGRCTNNB1
SCHEMBL2320678 0.83 MEN1 (0.33) HPGD
SCHEMBL2316423 0.82 BACE1 (0.38) HPGD
SCHEMBL2321527 0.81 IMPDH2 (0.31)
SCHEMBL2316316 0.81 AKR1B1 (0.36) AKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1609786-B1 5-alkenone-3,3-dimethyl-benzoxepines derivatives useful for the preparation of antidiabetic pentadienoic acids MERCK SANTE SAS (FR) 2011-08-03 EP claimed