SCHEMBL2319253

SCHEMBL2319253

COc1ccc2c(c1)C(CCC(C)=O)=CC(C)(C)CO2

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.43
NPC1 O15118 3/20 0.43
MAPT P10636 3/20 0.43
RAB9A P51151 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
LMNA P02545 2/20 0.43
TP53 P04637 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
MAOA P21397 1/20 0.43
SLC6A2 P23975 1/20 0.43
SLC6A3 Q01959 1/20 0.43
HTR2B P41595 2/20 0.38
SIGMAR1 Q99720 2/20 0.38
HTR1A P08908 1/20 0.38
ALDH1A1 P00352 2/20 0.38
GAA P10253 1/20 0.38
HPGD P15428 1/20 0.38
ALOX12 P18054 1/20 0.38
TDP1 Q9NUW8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2317591 0.91 CYP3A4 (0.43) KDM4ENPC1MAPTRAB9ASMN1; SMN2
SCHEMBL2316423 0.87 BACE1 (0.38) SMN1; SMN2HPGD
SCHEMBL14469715 0.86 HTR2B (0.34) KDM4ENPC1MAPTRAB9ASMN1; SMN2
SCHEMBL2316362 0.84 HTR1A (0.34) KDM4EMAPTSMN1; SMN2LMNACYP1A2
SCHEMBL2319041 0.83 CYP3A4 (0.35) KDM4ENPC1MAPTRAB9ASMN1; SMN2
SCHEMBL2322133 0.83 ALDH1A1 (0.39) KDM4EALDH1A1GAAHPGDCYP19A1
SCHEMBL2314396 0.83 MAPT (0.34) KDM4EMAPTCYP1A2CYP3A4ALDH1A1
SCHEMBL7031541 0.83 HTR2B (0.42) KDM4ENPC1MAPTRAB9ASMN1; SMN2
SCHEMBL2314339 0.82 PARP1 (0.38) KDM4ENPC1MAPTRAB9ASMN1; SMN2
SCHEMBL2320678 0.81 MEN1 (0.33) NPC1RAB9AHPGDMTNR1AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1609786-B1 5-alkenone-3,3-dimethyl-benzoxepines derivatives useful for the preparation of antidiabetic pentadienoic acids MERCK SANTE SAS (FR) 2011-08-03 EP claimed