SCHEMBL2314396

SCHEMBL2314396

CC(=O)CCC1=CC(C)(C)COc2ccc(Br)cc21

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.34
NR3C1 P04150 1/20 0.33
PGR P06401 1/20 0.33
AR P10275 1/20 0.33
APP P05067 6/20 0.32
CUL4A Q13619 1/20 0.32
CYP19A1 P11511 1/20 0.32
PBRM1 Q86U86 1/20 0.32
AKR1B1 P15121 1/20 0.31
MEN1 O00255 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
KMT2A Q03164 1/20 0.31
NPSR1 Q6W5P4 2/20 0.30
MAPK1 P28482 2/20 0.30
MITF O75030 1/20 0.30
HSP90AA1 P07900 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2316362 0.86 HTR1A (0.34) MAPTPGRCYP19A1MEN1CYP1A2
SCHEMBL2322133 0.85 ALDH1A1 (0.39) PGRARCYP19A1AKR1B1ALDH1A1
SCHEMBL2319689 0.85 NOTUM (0.34) MAPTPGRARCYP19A1AKR1B1
SCHEMBL2314339 0.84 PARP1 (0.38) MAPTMEN1CYP1A2CYP3A4KMT2A
SCHEMBL2320678 0.83 MEN1 (0.33) MEN1KMT2APTGS1PTGS2
SCHEMBL2319253 0.83 KDM4E (0.43) MAPTPGRCYP19A1CYP1A2CYP3A4
SCHEMBL2321527 0.81 IMPDH2 (0.31)
SCHEMBL2316316 0.81 AKR1B1 (0.36) AKR1B1
SCHEMBL2316423 0.80 BACE1 (0.38) CYP2C9
SCHEMBL2319041 0.78 CYP3A4 (0.35) MAPTNR3C1PGRARMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1609786-B1 5-alkenone-3,3-dimethyl-benzoxepines derivatives useful for the preparation of antidiabetic pentadienoic acids MERCK SANTE SAS (FR) 2011-08-03 EP claimed