SCHEMBL23257556

SCHEMBL23257556

C=CC(=O)Nc1cc(C(=O)NCC)cc(C(F)(F)F)c1

nearest known ligand 0.50

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TGM2 P21980 1/20 0.50
BCHE P06276 1/20 0.46
P2RX1 P51575 2/20 0.43
TRPA1 O75762 5/20 0.43
RHOC P08134 4/20 0.43
RHOA P61586 4/20 0.43
CYP1A2 P05177 1/20 0.43
CCR2 P41597 1/20 0.42
ALDH1A1 P00352 2/20 0.41
MAPT P10636 1/20 0.41
POLB P06746 1/20 0.41
TACR1 P25103 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22446313 0.83 RHOC (0.47) TGM2BCHEP2RX1TRPA1RHOC
SCHEMBL23257554 0.82 TGM2 (0.45) TGM2BCHEP2RX1RHOCRHOA
SCHEMBL22446314 0.80 RHOC (0.45) TGM2BCHEP2RX1TRPA1RHOC
SCHEMBL13752959 0.80 TACR1 (0.56) RHOCRHOAALDH1A1POLBTACR1
SCHEMBL18763049 0.80 TGM2 (0.69) TGM2P2RX1ALDH1A1MAPTTACR1
SCHEMBL20857042 0.80 P2RX1 (0.62) TGM2P2RX1TRPA1RHOCRHOA
SCHEMBL18763027 0.79 RHOC (0.44) TGM2BCHEP2RX1RHOCRHOA
SCHEMBL23256742 0.79 RHOC (0.47) TGM2BCHEP2RX1TRPA1RHOC
SCHEMBL23257559 0.77 TGM2 (0.43) TGM2BCHEP2RX1RHOCRHOA
SCHEMBL18778619 0.76 TGM2 (0.59) TGM2P2RX1ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021076755-A1 AN ACTIVITY-GUIDE MAP OF ELECTROPHILE-CYSTEINE INTERACTIONS IN PRIMARY HUMAN IMMUNE CELLS THE SCRIPPS RESEARCH INSTITUTE (US) 2021-04-22 WO disclosed