SCHEMBL23339243

SCHEMBL23339243

CN(CCCCN1CCN(c2ccc([N+](=O)[O-])cc2)CC1)c1ccccc1OC=O

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 4/20 0.47
HTR7 P34969 3/20 0.46
HTR2A P28223 2/20 0.44
HTR2C P28335 2/20 0.44
ADRA1D P25100 1/20 0.43
ADRA1A P35348 1/20 0.43
ADRA1B P35368 1/20 0.43
SIRT6 Q8N6T7 1/20 0.43
POLB P06746 1/20 0.42
ALDH1A1 P00352 1/20 0.42
LMNA P02545 1/20 0.42
MAPT P10636 1/20 0.42
DRD2 P14416 1/20 0.42
DRD4 P21917 1/20 0.42
DRD3 P35462 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23339729 0.87 HTR7 (0.48) HTR1AHTR7HTR2ADRD2DRD4
SCHEMBL23339699 0.79 DRD4 (0.46) HTR1AHTR7HTR2AMAPTDRD2
SCHEMBL23339235 0.79 DRD2 (0.37) HTR7HTR2AHTR2CALDH1A1DRD2
SCHEMBL23339232 0.75 ABCB1 (0.47)
SCHEMBL4507337 0.74 SIRT6 (0.60) HTR1AHTR7HTR2AHTR2CSIRT6
SCHEMBL19926115 0.73 HTR1A (0.58) HTR1ASIRT6POLBLMNAMAPT
SCHEMBL23339773 0.73 HTR1A (0.43) HTR1AHTR7HTR2ADRD2DRD3
SCHEMBL12005663 0.72 SIRT6 (0.63) HTR1AHTR7SIRT6POLBALDH1A1
SCHEMBL2730000 0.71 KDM4E (0.63) HTR1ASIRT6POLBALDH1A1LMNA
SCHEMBL6945690 0.71 SIRT6 (0.65) HTR1AHTR7SIRT6POLBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3102204-B1 HIGHLY SELECTIVE SIGMA 1 RECEPTOR LIGANDS AND RADIOLIGANDS AS PROBES IN NOCICEPTIVE PROCESSING AND THE PATHOPHYSIOLOGICAL STUDY OF MEMORY DEFICITS AND COGNITIVE DISORDERS THE UNIV OF MISSISSIPPI (US) 2021-05-05 EP disclosed