SCHEMBL23354512

SCHEMBL23354512

Cc1ncn(C)c1C(=O)CNC(=O)O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APOBEC3A P31941 4/20 0.38
APOBEC3G Q9HC16 3/20 0.38
EGLN1 Q9GZT9 1/20 0.37
ADORA2B P29275 2/20 0.33
MAPT P10636 1/20 0.33
THRB P10828 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.32
CTDSP1 Q9GZU7 1/20 0.31
BCAT2 O15382 2/20 0.31
LMNA P02545 1/20 0.31
HPGD P15428 1/20 0.31
FLT1 P17948 2/20 0.31
NPC1 O15118 1/20 0.31
TP53 P04637 1/20 0.31
RAB9A P51151 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
CYP2C19 P33261 1/20 0.31
KDR P35968 1/20 0.30
GDA Q9Y2T3 1/20 0.30
KDM4E B2RXH2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24927744 0.81 DYRK1A (0.38) MAPTL3MBTL1LMNAHPGDKDM4E
SCHEMBL25457959 0.79 APOBEC3A (0.46) APOBEC3AAPOBEC3GMAPTTHRBCTDSP1
SCHEMBL23367000 0.77 APOBEC3A (0.41) APOBEC3AAPOBEC3GMAPTCTDSP1BCAT2
SCHEMBL23354271 0.77 EGLN1 (0.40) APOBEC3AAPOBEC3GEGLN1ADORA2BMAPT
SCHEMBL3054669 0.76 APOBEC3A (0.42) APOBEC3AAPOBEC3GADORA2BCTDSP1BCAT2
Hydrochloric Acid SCHEMBL23354063 0.76 APOBEC3A (0.40) APOBEC3AAPOBEC3GMAPTCTDSP1HPGD
SCHEMBL23716719 0.74 APOBEC3A (0.41) APOBEC3AAPOBEC3GADORA2BCTDSP1BCAT2
SCHEMBL20360594 0.74 KDM4E (0.49) APOBEC3AAPOBEC3GMAPTTHRBL3MBTL1
SCHEMBL23354122 0.70 PREP (0.41) EGLN1LMNACYP2C19
SCHEMBL23354046 0.70 LMNA (0.38) APOBEC3AMAPTLMNAHPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4058448-B1 HYDANTOIN DERIVATIVES AS ADAMTS7 ANTAGONISTS FOR THE TREATMENT OF CARDIOVASCULAR DISEASES BAYER AG (DE) 2024-05-29 EP disclosed
US-20230027346-A1 SUBSTITUTED HYDANTOINAMIDES AS ADAMTS7 ANTAGONISTS BAYER AKTIENGESELLSCHAFT (DE) 2023-01-26 US disclosed
EP-4058448-A1 SUBSTITUTED HYDANTOINAMIDES AS ADAMTS7 ANTAGONISTS Bayer Aktiengesellschaft (DE) 2022-09-21 EP disclosed
WO-2021094436-A1 SUBSTITUTED HYDANTOINAMIDES AS ADAMTS7 ANTAGONISTS BAYER AKTIENGESELLSCHAFT (DE) 2021-05-20 WO disclosed
EP-3822268-A1 SUBSTITUTED HYDANTOINAMIDES AS ADAMTS7 ANTAGONISTS Bayer Aktiengesellschaft (DE) 2021-05-19 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230027346-A1 SUBSTITUTED HYDANTOINAMIDES AS ADAMTS7 ANTAGONISTS ADAMTS7, MMP7, ADAM17 APOBEC3A 545/4885APOBEC3G 602/4885EGLN1 449/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.