SCHEMBL2335629

SCHEMBL2335629

CCOC(=O)N(c1ccccc1Cl)c1c(C)noc1-c1ccc(-c2ccccc2C(=O)OC)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 4/20 0.44
SLC6A4 P31645 3/20 0.44
ALDH1A1 P00352 5/20 0.39
HPGD P15428 2/20 0.39
ACR P10323 1/20 0.39
FTO Q9C0B1 1/20 0.38
LTB4R2 Q9NPC1 1/20 0.38
KDM4E B2RXH2 3/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
AGTR1 P30556 1/20 0.36
AGTR2 P50052 1/20 0.36
BDKRB1 P46663 3/20 0.36
SLC6A2 P23975 1/20 0.36
TSHR P16473 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
HSD17B10 Q99714 1/20 0.35
MAPT P10636 3/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3709682 0.92 FTO (0.39) SLC6A3SLC6A4ALDH1A1HPGDACR
SCHEMBL2336114 0.91 LTB4R2 (0.37) ALDH1A1HPGDACRFTOLTB4R2
SCHEMBL3711509 0.84 ACR (0.36) ALDH1A1HPGDACRFTOKDM4E
SCHEMBL2332523 0.84 MAPT (0.40) ALDH1A1HPGDACRFTOKDM4E
SCHEMBL2342592 0.84 LPAR1 (0.39) SLC6A3SLC6A4ALDH1A1HPGDSLC6A2
SCHEMBL3711309 0.83 FTO (0.36) ALDH1A1HPGDACRFTOLTB4R2
SCHEMBL2336634 0.83 LPAR1 (0.43) ALDH1A1HPGDACRFTOKDM4E
SCHEMBL2335317 0.82 LPAR1 (0.38) ALDH1A1HPGDKDM4ESMN1; SMN2MEN1
SCHEMBL3714395 0.81 NR1H4 (0.40) ALDH1A1HPGDACRFTOSMN1; SMN2
SCHEMBL3704916 0.81 ALDH1A1 (0.41) ALDH1A1HPGDACRFTOKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2358688-A2 ANTAGONISTS OF LYSOPHOSPHATIDIC ACID RECEPTORS Amira Pharmaceuticals, Inc. (US) 2011-08-24 EP disclosed
WO-2010077882-A2 ANTAGONISTS OF LYSOPHOSPHATIDIC ACID RECEPTORS AMIRA PHARMACEUTICALS, INC. (US) 2010-07-08 WO disclosed
WO-2010077883-A2 ANTAGONISTS OF LYSOPHOSPHATIDIC ACID RECEPTORS AMIRA PHARMACEUTICALS, INC. (US) 2010-07-08 WO disclosed