SCHEMBL23367252

SCHEMBL23367252

O=Cc1cnn(-c2ccc(C(F)(F)F)cc2)n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.40
HIF1A Q16665 1/20 0.38
XDH P47989 1/20 0.35
HDAC1 Q13547 2/20 0.34
TDP1 Q9NUW8 1/20 0.34
MAPT P10636 1/20 0.33
ATM Q13315 1/20 0.33
ADRB2 P07550 1/20 0.33
ADRB1 P08588 1/20 0.33
ADRB3 P13945 1/20 0.33
NPBWR1 P48145 2/20 0.33
GSK3A P49840 1/20 0.33
GSK3B P49841 1/20 0.33
MCHR1 Q99705 1/20 0.32
KDM4E B2RXH2 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
CYP2C9 P11712 1/20 0.32
PTGS2 P35354 1/20 0.32
TRPV1 Q8NER1 1/20 0.32
CA12 O43570 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12442424 0.81 P2RX7 (0.42) P2RX7HDAC1MAPTKDM4EPTGS2
SCHEMBL11691729 0.78 P2RX7 (0.42) P2RX7MAPTATMKDM4EPTGS2
SCHEMBL11696173 0.78 P2RX7 (0.42) P2RX7HIF1AMAPTKDM4ENPSR1
SCHEMBL23367193 0.78 KIF11 (0.42) P2RX7
SCHEMBL9814514 0.78 P2RX7 (0.62) P2RX7HDAC1MAPTATMKDM4E
SCHEMBL23384990 0.75 MAPT (0.38) HIF1AXDHTDP1MAPTATM
SCHEMBL11766757 0.74 HTT (0.47) P2RX7HIF1AMAPTNPBWR1MCHR1
SCHEMBL11695053 0.74 P2RX7 (0.46) P2RX7XDHTDP1MAPTKDM4E
SCHEMBL9213953 0.74 GABRB3 (0.43)
SCHEMBL15578585 0.73 SRD5A2 (0.41) HIF1AHDAC1MAPTATMKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3822265-A1 SUBSTITUTED HYDANTOINAMIDES AS ADAMTS7 ANTAGONISTS Bayer AG (DE) 2021-05-19 EP disclosed