SCHEMBL23367473

SCHEMBL23367473

CNC(=O)NC(C=O)(CNC(=O)c1cnn(-c2ccccc2)n1)C(C)C

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 5/20 0.49
ADAMTS7 Q9UKP4 3/20 0.41
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
NTRK1 P04629 1/20 0.38
NTRK2 Q16620 1/20 0.38
CTSL P07711 1/20 0.35
ADORA2A P29274 2/20 0.35
IRAK4 Q9NWZ3 1/20 0.35
P2RX7 Q99572 1/20 0.34
LSS P48449 1/20 0.34
HDAC3 O15379 1/20 0.33
HDAC4 P56524 1/20 0.33
HDAC7 Q8WUI4 1/20 0.33
HDAC2 Q92769 1/20 0.33
HDAC8 Q9BY41 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
HDAC9 Q9UKV0 1/20 0.33
HDAC5 Q9UQL6 1/20 0.33
ADORA1 P30542 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6464483 0.74 HDAC1 (0.55) HDAC1ADAMTS7NPC1RAB9ANTRK1
SCHEMBL23367305 0.72 HDAC1 (0.43) HDAC1ADAMTS7NPC1RAB9ANTRK1
SCHEMBL23367625 0.70 ADAMTS7 (0.46) HDAC1ADAMTS7
SCHEMBL23384731 0.69 ADAMTS7 (0.41) HDAC1ADAMTS7NPC1RAB9ANTRK1
SCHEMBL23367557 0.68 ADAMTS7 (0.46) HDAC1ADAMTS7NPC1RAB9A
SCHEMBL23385052 0.68 ADAMTS7 (0.41) HDAC1ADAMTS7NPC1RAB9ANTRK1
SCHEMBL24938697 0.65 ADAMTS7 (0.57) HDAC1ADAMTS7NPC1RAB9ANTRK1
SCHEMBL23354910 0.65 ADAMTS7 (0.65) HDAC1ADAMTS7NPC1RAB9A
SCHEMBL29874194 0.65 ADAMTS7 (0.65) HDAC1ADAMTS7NPC1RAB9A
SCHEMBL1752087 0.64 P2RX7 (0.53) HDAC1ADAMTS7NPC1RAB9ANTRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3822265-A1 SUBSTITUTED HYDANTOINAMIDES AS ADAMTS7 ANTAGONISTS Bayer AG (DE) 2021-05-19 EP disclosed