SCHEMBL234576

SCHEMBL234576

N[C@]1(C(=O)O)[C@H]2[C@@H](C[C@H]1OCc1ccc(Cl)c(Cl)c1)[C@]2(F)C(=O)O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 4/20 1.00
GRM3 Q14832 4/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12273714 0.94 GRM2 (0.88) GRM2GRM3
SCHEMBL11886412 0.91 GRM2 (0.83) GRM2GRM3
SCHEMBL232371 0.91 GRM2 (0.83) GRM2GRM3
Hydrochloric Acid SCHEMBL232370 0.90 GRM2 (0.81) GRM2GRM3
SCHEMBL30120557 0.89 GRM2 (0.81) GRM2GRM3
SCHEMBL4964584 0.89 GRM2 (0.80) GRM2GRM3
SCHEMBL5961906 0.89 GRM2 (0.80) GRM2GRM3
SCHEMBL7070920 0.89 GRM2 (0.80) GRM2GRM3
SCHEMBL231526 0.89 GRM2 (0.80) GRM2GRM3
SCHEMBL2002949 0.88 GRM2 (0.79) GRM2GRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 103 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240335430-A1 Combination Therapy for Treating or Preventing Depression or Other Mood Diseases UNIV YALE (US) 2024-10-10 US claimed
US-20240240152-A1 Protection of Beta Cells from Immune Attack JOSLIN DIABETES CENTER (US) 2024-07-18 US claimed
US-20240033254-A1 Combination Therapy for Treating or Preventing Depression or Other Mood Diseases UNIV YALE (US) 2024-02-01 US claimed
CN-116267014-A Cyclic deuterated gaboxadol and its use for treating psychotic disorders CERTEGO治疗公司 2023-06-20 CN claimed
US-20230183238-A1 RING DEUTERATED GABOXADOL AND ITS USE FOR THE TREATMENT OF PSYCHIATRIC DISORDERS CERTEGO ABC, LLC 2023-06-15 US claimed
EP-4153549-A2 RING DEUTERATED GABOXADOL AND ITS USE FOR THE TREATMENT OF PSYCHIATRIC DISORDERS Certego Therapeutics Inc. (US) 2023-03-29 EP claimed
US-11597726-B2 Ring deuterated gaboxadol and its use for the treatment of psychiatric disorders Certego Therapeutics Inc. (US) 2023-03-07 US claimed
US-20220127261-A1 RING DEUTERATED GABOXADOL AND ITS USE FOR THE TREATMENT OF PSYCHIATRIC DISORDERS CERTEGO ABC, LLC 2022-04-28 US claimed
US-20210251969-A1 Combination Therapy for Treating or Preventing Depression or Other Mood Diseases YALE UNIVERSITY 2021-08-19 US claimed
EP-3129065-B1 TARGETED DRUG DELIVERY THROUGH AFFINITY BASED LINKERS AKAMARA THERAPEUTICS INC (US) 2026-05-13 EP disclosed
US-20260125651-A1 Protection of Beta Cells from Immune Attack JOSLIN DIABETES CENTER (US) 2026-05-07 US disclosed
US-20260098030-A1 NEGATIVE ALLOSTERIC MODULATORS OF METABOTROPIC GLUTAMATE RECEPTOR 2 UNIV VANDERBILT (US) 2026-04-09 US disclosed
US-12545895-B2 Protection of beta cells from immune attack JOSLIN DIABETES CENTER (US) 2026-02-10 US disclosed
EP-4673136-A1 NEGATIVE ALLOSTERIC MODULATORS OF METABOTROPIC GLUTAMATE RECEPTOR 2 Vanderbilt University (US) 2026-01-07 EP disclosed
US-20070021394-A1 2-Aminobicyclo[3.1.0]hexane-2,6-dicarboxylic ester derivative TAISHO PHARMACEUTICAL CO., LTD. (JP) 2007-01-25 US disclosed
US-20070021394-A1 2-Aminobicyclo[3.1.0]hexane-2,6-dicarboxylic ester derivative TAISHO PHARMACEUTICAL CO., LTD. (JP) 2007-01-25 US disclosed
US-7157594-B2 6-Fluorobicyclo[3.1.0]hexane derivatives TAISHO PHARMACEUTICAL CO., LTD. (JP) 2007-01-02 US disclosed
EP-1637517-A1 2-AMINOBICYCLO 3.1.0 HEXANE-2,6-DICARBOXYLIC ESTER DERIVATIVE Taisho Pharmaceutical Co. Ltd. (JP) 2006-03-22 EP disclosed
US-20050119345-A1 6-Fluorobicyclo[3.1.0]hexane derivatives TAISHO PHARMACEUTICAL CO., LTD. (JP) 2005-06-02 US disclosed
CN-1610557-A 6-fluorobicyclo [3.1.0] hexane derivatives TAISHO PHARMACEUTICAL CO LTD (JP) 2005-04-27 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050119345-A1 6-Fluorobicyclo[3.1.0]hexane derivatives GRM1, GRM2, GRM6 GRM2 2/4885GRM3 4/4885
US-20260098030-A1 NEGATIVE ALLOSTERIC MODULATORS OF METABOTROPIC GLUTAMATE RECEPTOR 2 GRM2, GRM1, GRIN2C GRM2 1/4885GRM3 5/4885
US-20230183238-A1 RING DEUTERATED GABOXADOL AND ITS USE FOR THE TREATMENT OF PSYCHIATRIC DISORDERS GABRD, GABRA6, GABRA3 GRM2 53/4885GRM3 29/4885
US-20070021394-A1 2-Aminobicyclo[3.1.0]hexane-2,6-dicarboxylic ester derivative GRIN2C, GRIK4, GRIN2B GRM2 13/4885GRM3 10/4885
US-20260125651-A1 Protection of Beta Cells from Immune Attack IAPP, SPPL2B, TXNL1 GRM2 4721/4885GRM3 4636/4885
US-12545895-B2 Protection of beta cells from immune attack PLIN1, GLS, GCKR GRM2 8/4885GRM3 32/4885
US-20220127261-A1 RING DEUTERATED GABOXADOL AND ITS USE FOR THE TREATMENT OF PSYCHIATRIC DISORDERS GABRD, GABRA6, GABRA3 GRM2 53/4885GRM3 29/4885
US-11597726-B2 Ring deuterated gaboxadol and its use for the treatment of psychiatric disorders GABRD, GABRA6, GABRA3 GRM2 53/4885GRM3 29/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.