SCHEMBL2346348

SCHEMBL2346348

NC(=O)CN(c1ccccc1)C1CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.47
HTT P42858 2/20 0.42
TAAR1 Q96RJ0 1/20 0.42
MITF O75030 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
KDM4E B2RXH2 1/20 0.41
MEN1 O00255 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
KMT2A Q03164 1/20 0.41
PAX8 Q06710 1/20 0.41
ALOX15 P16050 1/20 0.39
SIGMAR1 Q99720 2/20 0.37
HPGD P15428 1/20 0.37
NPSR1 Q6W5P4 1/20 0.36
DRD2 P14416 1/20 0.36
HTR2A P28223 1/20 0.36
HTR2C P28335 1/20 0.36
HTR2B P41595 1/20 0.36
LMNA P02545 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7371438 0.92 MEN1 (0.51) ALDH1A1HTTMITFSMN1; SMN2KDM4E
SCHEMBL5725403 0.86 ALDH1A1 (0.43) ALDH1A1SIGMAR1CHRM2CHRM3ADRA1A
SCHEMBL2037132 0.85 ALDH1A1 (0.51) ALDH1A1HTTTAAR1MITFSMN1; SMN2
SCHEMBL16335464 0.83 HTT (0.44) ALDH1A1HTTTAAR1MITFSMN1; SMN2
SCHEMBL2340823 0.78 ALDH1A1 (0.43) ALDH1A1HTTTAAR1MITFSMN1; SMN2
SCHEMBL3402515 0.78 OPRM1 (0.44) ALDH1A1HTTTAAR1MITFSMN1; SMN2
SCHEMBL3409354 0.74 HDAC1 (0.45) ALDH1A1HTTSMN1; SMN2MEN1NPC1
SCHEMBL11344206 0.74 KMT2A (0.48) ALDH1A1HTTMITFSMN1; SMN2KDM4E
SCHEMBL3404199 0.74 MEN1 (0.49) ALDH1A1HTTMITFSMN1; SMN2KDM4E
SCHEMBL11671526 0.73 KDM4E (0.50) ALDH1A1HTTMITFSMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2177502-A1 Compounds and their use Oryzon Genomics, S.A. (ES) 2010-04-21 EP claimed
EP-3397616-B1 LSD1 INHIBITORS MIRATI THERAPEUTICS INC (US) 2020-06-10 EP disclosed
EP-3105219-B9 CYCLOPROPYLAMINES AS LSD1 INHIBITORS INCYTE CORP (US) 2018-10-03 EP disclosed
EP-2361242-B1 OXIDASE INHIBITORS AND THEIR USE ORYZON GENOMICS SA (ES) 2018-08-01 EP disclosed
EP-3105219-B1 CYCLOPROPYLAMINES AS LSD1 INHIBITORS INCYTE CORP (US) 2018-04-11 EP disclosed
US-8524717-B2 Oxidase inhibitors and their use ORYZON GENOMICS, S.A. (ES) 2013-09-03 US disclosed
US-8524717-B2 Oxidase inhibitors and their use ORYZON GENOMICS, S.A. (ES) 2013-09-03 US disclosed
US-20110263604-A1 Oxidase inhibitors and their use ORYZON GENOMICS, S.A. (ES) 2011-10-27 US disclosed
US-20110263604-A1 Oxidase inhibitors and their use ORYZON GENOMICS, S.A. (ES) 2011-10-27 US disclosed
EP-2361242-A1 OXIDASE INHIBITORS AND THEIR USE Oryzon Genomics, S.A. (ES) 2011-08-31 EP disclosed
EP-2361242-A1 OXIDASE INHIBITORS AND THEIR USE Oryzon Genomics, S.A. (ES) 2011-08-31 EP disclosed
WO-2010043721-A1 OXIDASE INHIBITORS AND THEIR USE ORYZON GENOMICS, S.A. (ES) 2010-04-22 WO disclosed
WO-2010043721-A1 OXIDASE INHIBITORS AND THEIR USE ORYZON GENOMICS, S.A. (ES) 2010-04-22 WO disclosed
EP-2177502-A1 Compounds and their use Oryzon Genomics, S.A. (ES) 2010-04-21 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110263604-A1 Oxidase inhibitors and their use MAOA, PNPO, MAOB ALDH1A1 127/4885HTT 2541/4885TAAR1 919/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.