SCHEMBL2348652

SCHEMBL2348652

C=C(Br)Cc1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES1 P23141 3/20 0.50
CES2 O00748 2/20 0.50
AKR1B1 P15121 1/20 0.50
ALDH1A1 P00352 3/20 0.43
TSHR P16473 2/20 0.43
TRPA1 O75762 1/20 0.43
KMT2A Q03164 2/20 0.43
MEN1 O00255 1/20 0.43
HDAC8 Q9BY41 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
FNTA P49354 1/20 0.41
FNTB P49356 1/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
CALM1 P0DP23 1/20 0.41
TDP1 Q9NUW8 2/20 0.40
MAPK1 P28482 1/20 0.40
CTBP2 P56545 1/20 0.40
EPHX2 P34913 1/20 0.40
LMNA P02545 1/20 0.39
GAA P10253 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6187432 1.00 CES1 (0.50) CES1CES2AKR1B1ALDH1A1TSHR
SCHEMBL17708570 0.78 CES1 (0.55) CES1CES2AKR1B1ALDH1A1TSHR
SCHEMBL2241627 0.78 CES1 (0.55) CES1CES2AKR1B1ALDH1A1TSHR
SCHEMBL822099 0.78 CES1 (0.55) CES1CES2AKR1B1ALDH1A1TSHR
SCHEMBL12095508 0.78 CES1 (0.55) CES1CES2AKR1B1ALDH1A1TSHR
SCHEMBL31208444 0.77 CES1 (0.67) CES1CES2AKR1B1ALDH1A1TSHR
SCHEMBL5610463 0.77 CES1 (0.54) CES1CES2AKR1B1ALDH1A1TSHR
SCHEMBL1333665 0.76 CES1 (0.52) CES1CES2AKR1B1ALDH1A1TSHR
Ammonia Solution, Strong SCHEMBL574785 0.76 CES1 (0.52) CES1CES2AKR1B1ALDH1A1TSHR
SCHEMBL3855307 0.76 CES1 (0.52) CES1CES2AKR1B1ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109232422-B Preparation method of celecoxib 烟台万润药业有限公司 2020-07-07 CN claimed
CN-109232422-A A kind of preparation method of celecoxib 烟台万润药业有限公司 2019-01-18 CN claimed
CN-111484453-B Synthesis method of celecoxib 福建海西新药创制股份有限公司 2023-05-05 CN disclosed
CN-111484453-A Synthesis method of celecoxib 福建海西新药创制有限公司 2020-08-04 CN disclosed
CN-109232422-B Preparation method of celecoxib 烟台万润药业有限公司 2020-07-07 CN disclosed
CN-109232422-B Preparation method of celecoxib 烟台万润药业有限公司 2020-07-07 CN disclosed
US-10266503-B1 Sulfoxide ligand metal catalyzed oxidation of olefins THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 2019-04-23 US disclosed
CN-109232422-A A kind of preparation method of celecoxib 烟台万润药业有限公司 2019-01-18 CN disclosed
CN-109232422-A A kind of preparation method of celecoxib 烟台万润药业有限公司 2019-01-18 CN disclosed
WO-2013122364-A2 COMPOUND FOR ORGANIC ELECTRICAL ELEMENT, ORGANIC ELECTRICAL ELEMENT COMPRISING SAME, AND ELECTRONIC DEVICE THEREWITH 덕산하이메탈(주) (KR) 2013-08-22 WO disclosed
US-20110190137-A1 METHOD TO INHIBIT ETHYLENE RESPONSES IN PLANTS JACOBSON RICHARD MARTIN 2011-08-04 US disclosed
US-7296576-B2 Polymers for enhanced solubility of nanomaterials, compositions and methods therefor ZYVEX PERFORMANCE MATERIALS, LLC (US) 2007-11-20 US disclosed
US-20060041104-A1 Polymers for enhanced solubility of nanomaterials, compositions and methods therefor ZYVEX CORPORATION (US) 2006-02-23 US disclosed
EP-1409440-A4 A METHOD TO INHIBIT ETHYLENE RESPONSES IN PLANTS ROHM & HAAS (US) 2005-09-14 EP disclosed
US-20050065033-A1 Method to inhibit ethylene responses in plants JACOBSON RICHARD MARTIN (US) 2005-03-24 US disclosed
EP-1409440-A1 A METHOD TO INHIBIT ETHYLENE RESPONSES IN PLANTS ROHM AND HAAS COMPANY (US) 2004-04-21 EP disclosed
WO-2002068367-A1 A METHOD TO INHIBIT ETHYLENE RESPONSES IN PLANTS ROHM AND HAAS COMPANY (US) 2002-09-06 WO disclosed
US-4594467-A DEHYDROBROMINATING ALPH-BROMO-3,5-DICHLORO CUMENE WITH ALKALI METAL HYDROXIDE IN PRESENCE OF PHASE TRANSFER CATALYST BAYER AKTIENGESELLSCHAFT (DE) 1986-06-10 US disclosed
US-4446076-A Method of preparing 1,2-dibromo-2-cyano-(substituted)-alkane antimicrobial compounds MERCK & CO., INC. (US) 1984-05-01 US disclosed
US-4366170-A 1,2-Dibromo-2-cyano-2-(aryl)ethane(propane) antimicrobial compounds MERCK & CO., INC. (US) 1982-12-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050065033-A1 Method to inhibit ethylene responses in plants ERN1, CTH, CBS CES1 820/4885CES2 191/4885AKR1B1 2087/4885
US-20110190137-A1 METHOD TO INHIBIT ETHYLENE RESPONSES IN PLANTS ERN1, CTH, CBR3 CES1 721/4885CES2 154/4885AKR1B1 2037/4885
US-10266503-B1 Sulfoxide ligand metal catalyzed oxidation of olefins YAP1, ICOSLG, SPIN3 CES1 4488/4885CES2 4184/4885AKR1B1 2173/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.