SCHEMBL2348993

SCHEMBL2348993

Cc1ccc(C=O)nc1C(=O)O

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 1/20 0.42
ALDH1A1 P00352 4/20 0.36
MAPT P10636 3/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
PIN1 Q13526 1/20 0.35
TERT O14746 1/20 0.35
KDM4E B2RXH2 2/20 0.33
TDP1 Q9NUW8 2/20 0.33
RAB9A P51151 1/20 0.33
POLB P06746 1/20 0.33
APEX1 P27695 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
CYP3A4 P08684 1/20 0.33
RBP4 P02753 1/20 0.32
RRM2 P31350 1/20 0.32
HTT P42858 1/20 0.32
FGFR4 P22455 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2373944 0.75 ALDH1A1 (0.41) CCR1ALDH1A1MAPTSMN1; SMN2PIN1
SCHEMBL2222443 0.74 ALDH1A1 (0.40) ALDH1A1MAPTSMN1; SMN2PIN1KDM4E
SCHEMBL19857471 0.74 KDM4E (0.48) ALDH1A1MAPTSMN1; SMN2PIN1KDM4E
SCHEMBL3901458 0.73 GABRP (0.56) CCR1ALDH1A1SMN1; SMN2KDM4ETDP1
SCHEMBL6629423 0.73 CCR1 (0.50) CCR1ALDH1A1MAPTTERTRRM2
SCHEMBL847125 0.72 ALDH1A1 (0.39) ALDH1A1MAPTSMN1; SMN2PIN1KDM4E
SCHEMBL21332489 0.72 ALDH1A1 (0.39) ALDH1A1MAPTSMN1; SMN2PIN1KDM4E
SCHEMBL20475332 0.72 ALDH1A1 (0.39) ALDH1A1MAPTSMN1; SMN2PIN1KDM4E
SCHEMBL31715406 0.72 GABRP (0.55) ALDH1A1MAPTSMN1; SMN2PIN1KDM4E
SCHEMBL1428059 0.72 ALDH1A1 (0.46) ALDH1A1MAPTSMN1; SMN2PIN1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 25 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250082793-A1 MACROCYCLIC COMPOUNDS AND METHODS OF MAKING THE SAME JANSSEN BIOTECH, INC. 2025-03-13 US claimed
EP-4430040-A1 MACROCYCLIC COMPOUNDS AND METHODS OF MAKING THE SAME Janssen Biotech, Inc. (US) 2024-09-18 EP claimed
WO-2023084396-A1 MACROCYCLIC COMPOUNDS AND METHODS OF MAKING THE SAME JANSSEN BIOTECH, INC. (US) 2023-05-19 WO claimed
US-20250082793-A1 MACROCYCLIC COMPOUNDS AND METHODS OF MAKING THE SAME JANSSEN BIOTECH, INC. 2025-03-13 US disclosed
EP-4430040-A1 MACROCYCLIC COMPOUNDS AND METHODS OF MAKING THE SAME Janssen Biotech, Inc. (US) 2024-09-18 EP disclosed
EP-3318555-B1 BIFUNCTIONAL CHELATING AGENTS BWXT MEDICAL LTD (CA) 2023-08-16 EP disclosed
WO-2023084396-A1 MACROCYCLIC COMPOUNDS AND METHODS OF MAKING THE SAME JANSSEN BIOTECH, INC. (US) 2023-05-19 WO disclosed
EP-3318555-A1 BIFUNCTIONAL CHELATING AGENTS Nordion (Canada) Inc. (CA) 2018-05-09 EP disclosed
EP-2536691-B1 BIFUNCTIONAL CHELATING AGENTS Nordion (Canada) Inc (CA) 2017-11-22 EP disclosed
US-8772446-B2 Bifunctional chelating agents NORDION (CANADA) INC. (CA) 2014-07-08 US disclosed
EP-2536691-A1 BIFUNCTIONAL CHELATING AGENTS Nordion (Canada) Inc. (CA) 2012-12-26 EP disclosed
US-20080097119-A1 Disubstituted chalcone oximes having RARgamma retinoid receptor antagonist activity TSANG KWOK Y 2008-04-24 US disclosed
US-7253319-B2 Disubstituted chalcone oximes having RARγ retinoid receptor antagonist activity ALLERGAN, INC. (US) 2007-08-07 US disclosed
EP-1704139-A1 DISUBSTITUTED CHALCONE OXIMES AS SELECTIVE AGONISTS OF RAR y RETINOID RECEPTORS Allergan, Inc. (US) 2006-09-27 EP disclosed
EP-1701934-A2 DISUBSTITUTED CHALCONE OXIMES HAVING RAR(Gamma)-RETINOID RECEPTOR ANTAGONIST ACTIVITY Allergan, Inc. (US) 2006-09-20 EP disclosed
US-20050165095-A1 Disubstituted chalcone oximes having RARy retinoid receptor antagonist activity ALLERGAN, INC. 2005-07-28 US disclosed
WO-2005066116-A1 DISUBSTITUTED CHALCONE OXIMES AS SELECTIVE AGONISTS OF RARϜ RETINOID RECEPTORS ALLERGAN, INC. (US) 2005-07-21 WO disclosed
WO-2005066115-A2 DISUBSTITUTED CHALCONE OXIMES HAVING RARϜ RETINOID RECEPTOR ANTAGONIST ACTIVITY ALLERGAN, INC. (US) 2005-07-21 WO disclosed
US-20050148590-A1 Disubstituted chalcone oximes as selective agonists of RAR retinoid receptors ALLERGAN, INC. 2005-07-07 US disclosed
US-20050148623-A1 Prevent reproduct of aids virus ABBVIE INC. 2005-07-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050148623-A1 Prevent reproduct of aids virus SERPINB1, PRSS1, SERPINA3 CCR1 1559/4885ALDH1A1 1209/4885MAPT 1745/4885
US-20250082793-A1 MACROCYCLIC COMPOUNDS AND METHODS OF MAKING THE SAME PAICS, CD47, FURIN CCR1 106/4885ALDH1A1 2835/4885MAPT 1539/4885
US-20080097119-A1 Disubstituted chalcone oximes having RARgamma retinoid receptor antagonist activity RARG, RARB, RARA CCR1 890/4885ALDH1A1 421/4885MAPT 4778/4885
US-20050165095-A1 Disubstituted chalcone oximes having RARy retinoid receptor antagonist activity RARB, RARG, RARA CCR1 863/4885ALDH1A1 398/4885MAPT 4700/4885
US-20050148590-A1 Disubstituted chalcone oximes as selective agonists of RAR retinoid receptors RARG, RXRG, RARB CCR1 263/4885ALDH1A1 1103/4885MAPT 4165/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.