SCHEMBL23536225

SCHEMBL23536225

O=[N+]([O-])c1ccccc1N1CCC(CN2CCOCC2)CC1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CTSB P07858 1/20 0.49
CYP1A2 P05177 2/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C19 P33261 1/20 0.47
ALDH1A1 P00352 6/20 0.46
KMT2A Q03164 4/20 0.46
MEN1 O00255 2/20 0.46
HTT P42858 2/20 0.46
MAPT P10636 7/20 0.46
LMNA P02545 2/20 0.46
GAA P10253 2/20 0.46
NPSR1 Q6W5P4 1/20 0.46
TDP1 Q9NUW8 2/20 0.45
MAPK1 P28482 1/20 0.45
KDM4E B2RXH2 1/20 0.45
PKM P14618 2/20 0.44
HTR1A P08908 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29931897 1.00 CTSB (0.49) CTSBCYP1A2CYP2D6CYP2C19ALDH1A1
SCHEMBL23536471 0.84 HTT (0.48) CTSBALDH1A1KMT2AHTTMAPT
SCHEMBL29948611 0.84 HTT (0.48) CTSBALDH1A1KMT2AHTTMAPT
SCHEMBL30779614 0.82 CTSB (0.68) CTSBCYP1A2CYP2D6CYP2C19ALDH1A1
SCHEMBL2206983 0.82 CTSB (0.68) CTSBCYP1A2CYP2D6CYP2C19ALDH1A1
SCHEMBL29931922 0.82 ALDH1A1 (0.47) ALDH1A1KMT2AHTTMAPTLMNA
SCHEMBL23536258 0.82 ALDH1A1 (0.47) ALDH1A1KMT2AHTTMAPTLMNA
SCHEMBL3435490 0.81 CTSB (0.52) CTSBCYP1A2ALDH1A1KMT2AMEN1
SCHEMBL4939842 0.80 ALDH1A1 (0.56) CYP2C19ALDH1A1KMT2AMEN1MAPT
SCHEMBL28241 0.79 KMT2A (0.60) ALDH1A1KMT2AMEN1MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4076423-A1 TRPML MODULATORS Casma Therapeutics, Inc. (US) 2022-10-26 EP disclosed
CN-115087440-A TRPML modulators 卡斯玛治疗公司 2022-09-20 CN disclosed
WO-2021127337-A1 TRPML MODULATORS CASMA THERAPEUTICS, INC. (US) 2021-06-24 WO disclosed