SCHEMBL23536668

SCHEMBL23536668

Fc1cc(Cl)ccc1Oc1cccc2[nH]ncc12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 1/20 0.49
TRPA1 O75762 1/20 0.47
NOS1 P29475 5/20 0.46
RHEB Q15382 2/20 0.46
SLC6A2 P23975 2/20 0.44
SLC6A4 P31645 2/20 0.44
KCNH2 Q12809 1/20 0.44
SLC6A3 Q01959 1/20 0.44
P2RX3 P56373 1/20 0.42
AXL P30530 2/20 0.40
RAF1 P04049 2/20 0.40
BRAF P15056 2/20 0.40
DYRK1A Q13627 1/20 0.40
EPAS1 Q99814 2/20 0.39
EGFR P00533 1/20 0.39
ERBB2 P04626 1/20 0.39
CYP11B1 P15538 1/20 0.39
CYP11B2 P19099 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2877152 0.84 ROCK2 (0.54) ROCK2TRPA1NOS1AXLRAF1
SCHEMBL28199257 0.81 NOS1 (0.57) ROCK2NOS1AXLEPAS1
SCHEMBL2876576 0.79 HSPB1 (0.50) ROCK2TRPA1NOS1RAF1BRAF
SCHEMBL3484118 0.76 NOS1 (0.50) ROCK2NOS1RHEBP2RX3AXL
SCHEMBL28509646 0.74 NOS1 (0.48) TRPA1NOS1SLC6A2SLC6A4KCNH2
SCHEMBL30194080 0.74 NOS1 (0.48) TRPA1NOS1SLC6A2SLC6A4KCNH2
SCHEMBL23536624 0.73 NOS1 (0.53) TRPA1NOS1AXLRAF1BRAF
SCHEMBL17714209 0.71 CYP11B1 (0.54) TRPA1SLC6A2SLC6A4KCNH2SLC6A3
SCHEMBL5951586 0.69 AXL (0.63) TRPA1NOS1AXLRAF1BRAF
SCHEMBL30469214 0.69 AXL (0.63) TRPA1NOS1AXLRAF1BRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021127333-A1 TRPML MODULATORS CASMA THERAPEUTICS, INC. (US) 2021-06-24 WO disclosed