SCHEMBL2356597

SCHEMBL2356597

CCCCOC(=O)NC(Cc1ccc(-c2cccnc2)cc1)C(=O)O

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP19A1 P11511 1/20 0.51
CYP2C9 P11712 1/20 0.51
CYP2C19 P33261 1/20 0.51
MME P08473 2/20 0.50
ACE P12821 2/20 0.50
CPA1 P15085 2/20 0.50
ACE2 Q9BYF1 2/20 0.50
ITGB1 P05556 2/20 0.49
ITGA4 P13612 2/20 0.49
ITGB3 P05106 10/20 0.48
ITGAV P06756 4/20 0.48
L3MBTL1 Q9Y468 1/20 0.46
GPR132 Q9UNW8 1/20 0.46
PPARG P37231 1/20 0.46
FAAH O00519 1/20 0.46
ITGA2B P08514 6/20 0.46
MMP12 P39900 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3820286 0.89 GPR132 (0.52) CYP3A4ITGB1ITGA4ITGB3L3MBTL1
SCHEMBL5498526 0.89 GPR132 (0.52) CYP3A4ITGB1ITGA4ITGB3L3MBTL1
SCHEMBL2358936 0.89 MME (0.51) MMEACECPA1ACE2ITGB1
SCHEMBL9936982 0.89 MME (0.61) MMEACECPA1ACE2ITGB1
SCHEMBL15201783 0.89 MME (0.61) MMEACECPA1ACE2ITGB1
SCHEMBL4966319 0.84 ITGB3 (0.52) ACEACE2ITGB1ITGA4ITGB3
SCHEMBL7758997 0.83 ITGB3 (0.58) MMEACECPA1ACE2ITGB1
SCHEMBL2185240 0.83 ITGB3 (0.58) MMEACECPA1ACE2ITGB1
SCHEMBL844471 0.83 ITGB3 (0.58) MMEACECPA1ACE2ITGB1
SCHEMBL2312378 0.81 CTSS (0.58) CYP3A4MMEACEACE2ITGA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2350031-A2 MACROCYCLIC COMPOUNDS FOR INHIBITION OF TUMOR NECROSIS FACTOR ALPHA Ensemble Therapeutics Corporation (US) 2011-08-03 EP disclosed