SCHEMBL23601223

SCHEMBL23601223

CC(=O)Nc1ccc(-c2cccc(N(C)c3nc(=N)n(C=N)c4cc(N)ccc34)c2)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 2/20 0.38
DHODH Q02127 3/20 0.37
PARP1 P09874 2/20 0.37
BACE1 P56817 1/20 0.36
MTNR1A P48039 1/20 0.36
MTNR1B P49286 1/20 0.36
CHEK1 O14757 1/20 0.35
ALDH1A1 P00352 3/20 0.35
HPGD P15428 3/20 0.35
KDM4E B2RXH2 2/20 0.35
NPC1 O15118 1/20 0.35
TP53 P04637 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
HSD17B10 Q99714 1/20 0.35
HSD17B1 P14061 1/20 0.35
HSD17B2 P37059 1/20 0.35
HDAC1 Q13547 1/20 0.35
CSF1R P07333 1/20 0.35
FGFR1 P11362 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23601273 0.90 TDP1 (0.39) AOC3DHODHMTNR1AMTNR1BCHEK1
SCHEMBL23601197 0.82 MAPT (0.43) MTNR1AMTNR1BALDH1A1HPGDKDM4E
SCHEMBL23577153 0.81 AOC3 (0.38) AOC3DHODHPARP1BACE1MTNR1A
SCHEMBL29909552 0.81 AOC3 (0.38) AOC3DHODHPARP1BACE1MTNR1A
SCHEMBL23601707 0.76 PDE5A (0.42) DHODHKDR
SCHEMBL23601857 0.75 DHODH (0.35) DHODHALDH1A1HPGDKDM4ENPC1
SCHEMBL23601250 0.73 DHODH (0.33) DHODHMAPT
SCHEMBL23601374 0.73 DHODH (0.37) DHODHHPGDMAP4K4
SCHEMBL23600472 0.73 KDM4E (0.34) DHODHALDH1A1KDM4EMEN1MAPT
SCHEMBL23601587 0.73 EGFR (0.34) DHODHBACE1CHEK1ALDH1A1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021130638-A1 DIACYLGLYCEROL KINASE MODULATING COMPOUNDS CARNA BIOSCIENCES, INC. (JP) 2021-07-01 WO disclosed