SCHEMBL2361085

SCHEMBL2361085

COc1cc2[nH]c(-c3c(F)cccc3Cl)nc2cc1C#N

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
AMY1A P0DUB6 6/20 0.44
DGAT1 O75907 2/20 0.44
PTGES O14684 7/20 0.41
RHEB Q15382 1/20 0.41
JAK2 O60674 1/20 0.40
PDE7A Q13946 1/20 0.39
ORAI1 Q96D31 1/20 0.39
SRC P12931 1/20 0.38
HTR2A P28223 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2361888 0.80 AMY1A (0.47) AMY1ADGAT1PTGESJAK2PDE7A
SCHEMBL2362277 0.79 PLAU (0.51) AMY1ADGAT1
SCHEMBL2360991 0.77 RHEB (0.52) DGAT1PTGESRHEBJAK2
SCHEMBL2361306 0.76 AMY1A (0.44) AMY1ADGAT1PTGESPDE7AORAI1
SCHEMBL1512040 0.74 IDH1 (0.41) SRC
SCHEMBL2361250 0.74 AMY1A (0.43) AMY1ADGAT1PTGESJAK2PDE7A
SCHEMBL13405914 0.74 RHEB (0.54) AMY1ADGAT1PTGESRHEBJAK2
SCHEMBL2361475 0.74 DGAT1 (0.43) AMY1ADGAT1PTGESPDE7AORAI1
SCHEMBL2361209 0.73 PTGES (0.43) AMY1ADGAT1PTGESPDE7AORAI1
SCHEMBL2361234 0.73 PTGES (0.45) AMY1ADGAT1PTGESPDE7AORAI1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011099832-A2 NOVEL BENZIMIDAZOLE COMPOUND, PREPARATION METHOD THEREOF AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME CRYSTALGENOMICS, INC. (KR) 2011-08-18 WO disclosed
WO-2011099832-A2 NOVEL BENZIMIDAZOLE COMPOUND, PREPARATION METHOD THEREOF AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME CRYSTALGENOMICS, INC. (KR) 2011-08-18 WO disclosed