SCHEMBL2361289

SCHEMBL2361289

COC(=O)c1ccc2[nH]c(C(=O)Nc3ccc4[nH]c(-c5c(F)cccc5Cl)nc4c3)nc2c1

nearest known ligand 0.48

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 3/20 0.48
RHEB Q15382 1/20 0.46
PTGES O14684 3/20 0.45
MAPT P10636 3/20 0.43
NR2E3 Q9Y5X4 1/20 0.43
ATM Q13315 1/20 0.43
TP53 P04637 1/20 0.43
KDR P35968 1/20 0.42
MAOB P27338 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2362023 0.89 RHEB (0.57) DGAT1RHEBPTGESTP53
SCHEMBL2361142 0.86 DGAT1 (0.44) DGAT1RHEBPTGESMAPTNR2E3
SCHEMBL2361214 0.85 CSNK1E (0.52) DGAT1RHEBMAPTTP53
SCHEMBL2365435 0.84 PTGES (0.48) DGAT1PTGESMAPTNR2E3TP53
SCHEMBL2361026 0.83 DGAT1 (0.41) DGAT1RHEBPTGESMAPTNR2E3
SCHEMBL2361492 0.80 NR2E3 (0.64) DGAT1MAPTNR2E3TP53
SCHEMBL2361432 0.79 KDM4E (0.47) DGAT1RHEBPTGESMAPTTP53
SCHEMBL2362063 0.78 KDM4E (0.47) DGAT1RHEBPTGESMAPTTP53
SCHEMBL2361818 0.77 RAB9A (0.47) RHEBPTGESMAPTTP53
SCHEMBL2362094 0.77 PTGER4 (0.44) DGAT1PTGESMAPTNR2E3MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011099832-A2 NOVEL BENZIMIDAZOLE COMPOUND, PREPARATION METHOD THEREOF AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME CRYSTALGENOMICS, INC. (KR) 2011-08-18 WO disclosed